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Results for "

human SETDB1

" in MedChemExpress (MCE) Product Catalog:

2

Inhibitors & Agonists

2

Recombinant Proteins

1

Oligonucleotides

Cat. No. Product Name Target Research Areas Chemical Structure
  • HY-141539
    SETDB1-TTD-IN-1
    5 Publications Verification

    		 Histone Methyltransferase Akt Cancer
    SETDB1-TTD-IN-1 is a SETDB1 methyltransferase activator and SETDB1-TTD competitive inhibitor (Kd of 88 nM), and selectivity for SETDB1-TTD over other tudor and bromodomain proteins. SETDB1-TTD-IN-1 stimulates methyltransferase activity via increased catalytic activity, promotes Akt1 Lys64 methylation, Akt1 Thr308 phosphorylation and activation. SETDB1-TTD-IN-1 prevents SETDB1-TTD-histone H3 peptide association, induces global gene expression changes, exhibits cellular target engagement, and acts as a tool compound for SETDB1-TTD function exploration. SETDB1-TTD-IN-1 can be used for the research of breast cancer .
    SETDB1-TTD-IN-1
  • HY-RS12748
    SETDB1 Human Pre-designed siRNA Set A

    		Small Interfering RNA (siRNA) Others

    SETDB1 Human Pre-designed siRNA Set A contains three designed siRNAs for SETDB1 gene (Human), as well as a negative control, a positive control, and a FAM-labeled negative control.

    SETDB1 Human Pre-designed siRNA Set A
    SETDB1 Human Pre-designed siRNA Set A

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