34 Results for "

substrato pept

" in MedChemExpress (MCE) Product Catalog:
Products (34)

34 Results for "substrato pept" in MCE Product Catalog:

5
5 Cited Publications
Cat. No.: HY-B1190
CAS No.: 50370-12-2
Synonyms: BL-S 578
Target:  

Bacterial Antibiotic EAAT

Research Areas:  

Infection Neurological Disease

Cefadroxil is an orally active broad-spectrum cephalosporin antibiotic. Cefadroxil inhibits bacterial cell wall synthesis and enhances the expression of glutamate transporter-1. Cefadroxil is dependent on the intestinal peptide transporter PepT1 for small intestinal absorption. Cefadroxil has inhibitory and bactericidal activity against a variety of Gram-positive and Gram-negative bacteria and has analgesic effects on neuropathic pain .
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5
5 Cited Publications
Cat. No.: HY-B1190A
CAS No.: 66592-87-8
Synonyms: BL-S 578 hydrate
Target:  

Bacterial Antibiotic EAAT

Research Areas:  

Infection Neurological Disease

Cefadroxil hydrate is an orally active broad-spectrum cephalosporin antibiotic. Cefadroxil hydrate inhibits bacterial cell wall synthesis and enhances the expression of glutamate transporter-1. Cefadroxil hydrate is dependent on the intestinal peptide transporter PepT1 for small intestinal absorption. Cefadroxil hydrate has inhibitory and bactericidal activity against a variety of Gram-positive and Gram-negative bacteria and has analgesic effects on neuropathic pain .
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2
2 Cited Publications
Cat. No.: HY-111956B
CAS No.: 2703746-41-0
Purity:  98.77%
Target:  

Fluorescent Dye

Research Areas:  

Cancer

D-Ala-Lys-AMCA hydrochloride is a known proton-coupled oligopeptide transporter 1 (PEPT1) substrate that emits blue fluorescence. D-Ala-Lys-AMCA hydrochloride may be transported into liver cancer cells and Caco-2 cells based on fluorescence analysis. D-Ala-Lys-AMCA hydrochloride can be used for characterizing PEPT1-specific substrates or inhibitors (Ex/Em = 390/480 nm) .
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1
1 Cited Publications
Cat. No.: HY-B1258
CAS No.: 56-91-7
Synonyms: Aminomethylbenzoic acid; α-Amino-p-toluic acid
Research Areas:  

Cancer

4-(Aminomethyl)benzoic acid is a competitive inhibitor of PepT1 and has antifibrinolytic activity .
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1
1 Cited Publications
Cat. No.: HY-P704352
Purity:  ≥ 95%, as determined by reducing SDS-PAGE.
Synonyms: APP; PreA4; Prev. AD1; CVAP; Alzheimer Disease Amyloid A4 Protein Homolog; Beta-Amyloid Precursor Protein; Amyloid-Beta Precursor Protein; Testicular Tissue Protein Li 2; Amyloid Precursor Protein; Beta-Amyloid peptide(1-40); Alpha-SAPP; Beta-Amyloid pept
Species:  
Human
Source:  
HEK293
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Cat. No.: HY-W010162
CAS No.: 1948-31-8
Synonyms: L-Alanyl-L-alanine; Ala-Ala
H-Ala-Ala-OH is a substrate of human intestinal oligopeptide transporter (PEPT1/SLC15A1), with an IC50 of 0.25 mM and an EC50 of 0.08 mM against human PEPT1. When used as a dipeptide linker in antibody-drug conjugates (ADCs) loaded with glucocorticoid receptor regulator payloads, H-Ala-Ala-OH enables efficient intracellular payload release .
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Cat. No.: HY-Y1080
CAS No.: 19764-30-8
Synonyms: N-Acetyl-D-leucine
N-Acetyl-R-leucine is an amino-protecting group N-substituted chiral amino acid. N-Acetyl-R-leucine is a PepT1 and MCT1 inhibitor with IC50 of 0.74 and 11 mM, respectively. N-Acetyl-R-leucine can be used for LysoTracker signaling studies .
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Cat. No.: HY-W011165
CAS No.: 52123-30-5
Synonyms: L-Lysyl-L-lysine dihydrochloride
Lysyllysine dihydrochloride (L-Lysyl-L-lysine dihydrochloride) is an orally active PepT1 substrate. Lysyllysine dihydrochloride enhances whole-body protein synthesis, improves intestinal structure, alleviates intestinal mucosal inflammation, and exhibits higher lysine bioavailability in neonatal piglets with PN-induced intestinal atrophy. Lysyllysine dihydrochloride inhibits the growth of axenic cyanobacterial strains and induces their cell lysis. Lysyllysine dihydrochloride can be used in studies related to intestinal atrophy and metabolism .
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Cat. No.: HY-111956
CAS No.: 375822-19-8
Target:  

Fluorescent Dye

Research Areas:  

Cancer

D-Ala-Lys-AMCA is a known proton-coupled oligopeptide transporter 1 (PEPT1) substrate that emits blue fluorescence. D-Ala-Lys-AMCA may be transported into liver cancer cells and Caco-2 cells based on fluorescence analysis. D-Ala-Lys-AMCA can be used for characterizing PEPT1-specific substrates or inhibitors (Ex/Em = 390/480 nm) .
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Cat. No.: HY-W327145
CAS No.: 45234-02-4
Target:  

Endogenous Metabolite

Research Areas:  

Infection

Lysylglutamic acid is a dipeptide formed by combining two amino acids, Lysine (Lys) and Glutamic acid (Glu). The Ki value of the membrane transporter PEPT1 was 1.3 mM .
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Cat. No.: HY-B1190R
CAS No.: 50370-12-2
Synonyms: BL-S 578 (Standard)
Cefadroxil (Standard) is the analytical standard of Cefadroxil (HY-B1190). This product is intended for research and analytical applications. Cefadroxil is an orally active broad-spectrum cephalosporin antibiotic. Cefadroxil inhibits bacterial cell wall synthesis and enhances the expression of glutamate transporter-1. Cefadroxil is dependent on the intestinal peptide transporter PepT1 for small intestinal absorption. Cefadroxil has inhibitory and bactericidal activity against a variety of Gram-positive and Gram-negative bacteria and has analgesic effects on neuropathic pain .
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Cat. No.: HY-P4019
CAS No.: 121822-32-0
Target:  

HIV Protease

Research Areas:  

Others

Ac-Ser-Gln-Asn-Tyr-Pro-Val-Val-NH2 is a substrato peptídico of HIV-1 protease. Ac-Ser-Gln-Asn-Tyr-Pro-Val-Val-NH2 acts as the variable substrate in a peptidolytic assay to quantify the inhibition of the protease .
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Cat. No.: HY-W727334
CAS No.: 41745-47-5
Research Areas:  

Others

H-Glu-Pro-OH is a Xaa-Pro dipeptide with affinity for the intestinal H +/peptide cotransporter (PEPT1), with a Ki value of 0.26 mM .
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Cat. No.: HY-120791
CAS No.: 13184-13-9
Synonyms: L-Lysyl-L-lysine
Lysyllysine (L-Lysyl-L-lysine ) is an orally active PepT1 substrate. Lysyllysine enhances whole-body protein synthesis, improves intestinal structure, alleviates intestinal mucosal inflammation, and exhibits higher lysine bioavailability in neonatal piglets with PN-induced intestinal atrophy. Lysyllysine inhibits the growth of axenic cyanobacterial strains and induces their cell lysis. Lysyllysine can be used in studies related to intestinal atrophy and metabolism .
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Cat. No.: HY-B1190S
CAS No.: 1426174-38-0
Synonyms: BL-S 578-d4 hydrate
Cefadroxil-d4 (hydrate) is the deuterium labeled Cefadroxil hydrate (HY-B1190A). Cefadroxil hydrate is an orally active broad-spectrum cephalosporin antibiotic. Cefadroxil hydrate inhibits bacterial cell wall synthesis and enhances the expression of glutamate transporter-1. Cefadroxil hydrate is dependent on the intestinal peptide transporter PepT1 for small intestinal absorption. Cefadroxil hydrate has inhibitory and bactericidal activity against a variety of Gram-positive and Gram-negative bacteria and has analgesic effects on neuropathic pain .
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Cat. No.: HY-111956A
Target:  

Fluorescent Dye

Research Areas:  

Cancer

D-Ala-Lys-AMCA TFA is a known proton-coupled oligopeptide transporter 1 (PEPT1) substrate that emits blue fluorescence. D-Ala-Lys-AMCA TFA may be transported into liver cancer cells and Caco-2 cells based on fluorescence analysis. D-Ala-Lys-AMCA TFA can be used for characterizing PEPT1-specific substrates or inhibitors (Ex/Em = 390/480 nm) .
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Cat. No.: HY-B2072AR
CAS No.: 102039-86-1
Research Areas:  

Infection

Cefadroxil (hydrate) (Standard) is the analytical standard of Cefadroxil (hydrate). This product is intended for research and analytical applications. Cefadroxil hydrate (BL-S 578 hydrate) is an orally active and first-generation cephalosporin with a broad spectrum antibacterial activity. Cefadroxil hydrate (BL-S 578 hydrate) also acts as a substrate of the peptide transporter PEPT1 and PEPT2 .
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Cat. No.: HY-117110
CAS No.: 2418-69-1
Synonyms: H-Arg-Pro-OH
Target:  

Proton Pump

Research Areas:  

Metabolic Disease

Arginylproline (H-Arg-Pro-OH) is a dipeptide consisted of arginine and proline. Arginylproline reduces intracellular triglyceride (TG) levels stimulated by Oleic acid (HY-N1446), through the peptide transporter 1 (PepT1) pathway .
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Cat. No.: HY-B1258S
Synonyms: Aminomethylbenzoic acid-13C2,15N; α-Amino-p-toluic acid-13C2,15N
Intermediate of tranexamic Acid- 13C2, 15N (Aminomethylbenzoic acid- 13C2, 15N) is 13C and 15N labeled 4-(Aminomethyl)benzoic acid. 4-(Aminomethyl)benzoic acid is a competitive inhibitor of PepT1 and has antifibrinolytic activity .
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Cat. No.: HY-P4296
CAS No.: 57836-11-0
Research Areas:  

Others

H-Gly-Sar-Sar-OH is an orally active tripeptide. H-Gly-Sar-Sar-OH is transported through PepT1 within Caco-2 cells. H-Gly Sar Sar OH has potential applications in material transportation .
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