1. GPCR/G Protein
  2. LPL Receptor
  3. AS2717638

AS2717638 

Cat. No.: HY-114379
Handling Instructions

AS2717638 is an oral active and selective lysophosphatidic acid receptor 5 (LPA5) antagonist, with an IC50 of 38 nM for hLPA5. AS2717638 also significantly improves PGE2-, PGF-, and AMPA-induced allodynia.

For research use only. We do not sell to patients.

AS2717638 Chemical Structure

AS2717638 Chemical Structure

CAS No. : 2148339-28-8

Size Price Stock Quantity
10 mM * 1 mL in DMSO USD 495 In-stock
Estimated Time of Arrival: December 31
5 mg USD 450 In-stock
Estimated Time of Arrival: December 31
10 mg USD 750 In-stock
Estimated Time of Arrival: December 31
50 mg   Get quote  
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Based on 1 publication(s) in Google Scholar

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Description

AS2717638 is an oral active and selective lysophosphatidic acid receptor 5 (LPA5) antagonist, with an IC50 of 38 nM for hLPA5. AS2717638 also significantly improves PGE2-, PGF-, and AMPA-induced allodynia[1].

IC50 & Target

IC50: 38 nM (hLPA5)[1].

Molecular Weight

447.48

Formula

C₂₅H₂₅N₃O₅

CAS No.

2148339-28-8

SMILES

O=C1N(C2=NOC3=C2C=C(C)C=C3)C=C(C(N4CCCCC4)=O)C5=C1C=C(OC)C(OC)=C5

Shipping

Room temperature in continental US; may vary elsewhere

Storage
Powder -20°C 3 years
  4°C 2 years
In solvent -80°C 6 months
  -20°C 1 month
References
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AS2717638
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HY-114379
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