Drug Derivative
Drug derivative
Drug derivatives are derived from parent compounds. They replace or add atoms and groups through chemical reactions to optimize the various properties of the parent compound and reduce side effects. The application of drug derivatives provides a diverse compound library for drug research and development and accelerates the discovery of new drugs. For example, urea derivatives Glibenclamide can prolong the blood sugar-lowering effect of anti-diabetic drugs.
References:
- [1]. Vardanyan RS, et al. Fentanyl-related compounds and derivatives: current status and future prospects for pharmaceutical applications. Future Med Chem. 2014 Mar;6(4):385-412.x
- [2]. Ghosh AK, et al. Urea Derivatives in Modern Drug Discovery and Medicinal Chemistry. J Med Chem. 2020 Mar 26;63(6):2751-2788.x
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Drug Derivative Related Products (4032)
Related Products (4032)
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2,3-Dihydroxy-4-methoxybenzoic acid
0 Images2,3-Dihydroxy-4-methoxybenzoic acid is a Benzoic acid (HY-N0216) derivative that can be isolated from extracted from sweet cherry fruits (Prunus avium). 2,3-Dihydroxy-4-methoxybenzoic acid can be used as an organic synthesis intermediate used for the synthesis of active molecules.
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PPO-IN-22
0 ImagesCat. No.: HY-178165PPO-IN-22 (Compound B-04) is a benzothiazol-2(3H)-one derivative. PPO-IN-22 is a herbicide. PPO-IN-22 exhibits excellent post-emergence herbicidal activity against broadleaf weeds. PPO-IN-22 demonstrates potent pre-emergence activity against both dicotyledonous and monocotyledonous weeds. PPO-IN-22 exhibits favorable crop safety as a selective pre-emergence herbicide in soybean, peanut, and cotton cultivation systems.
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Tafluprost ethyl amide
0 ImagesTafluprost ethyl amide is a derivative of Tafluprost (HY-B0600). Tafluprost ethyl amide is commonly used in studies related to eyelash hypotrichosis, and it can also be applied in research related to the cosmetic field.
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1-Dodecanoyl-sn-glycerophosphoethanolamine
0 ImagesCat. No.: HY-165221CAS No.: 120578-22-51-Dodecanoyl-sn-glycerophosphoethanolamine, a derivative of phosphatidylethanolamine, interacts with Cinnamycin (HY-P1695) to induce conformational changes. 1-Dodecanoyl-sn-glycerophosphoethanolamine is applicable to studies related to antibiotic synthesis.
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PCPr hydrochloride
0 ImagesCat. No.: HY-W408972CAS No.: 1934-55-0PCPr (hydrochloride) is a compound derived from phencyclidine.
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Ethiofencarb-sulfoxide
0 ImagesCat. No.: HY-W714188CAS No.: 53380-22-6Ethiofencarb-sulfoxide is a pesticide metabolite.
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Nepinalone hydrochloride (Standard)
0 ImagesCat. No.: HY-106873ARCAS No.: 22443-55-6Nepinalone hydrochloride (Standard) is the analytical standard of Nepinalone (hydrochloride) (HY-106873A). This product is intended for research and analytical applications. Nepinalone hydrochloride, an alchilaminate derivative of β-tetralone and an orally active cough suppressant, possesses a non-opioid antitussive activity.
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N-(1,2-Dithiolane-3-pentanoyl)-Glu-Ala
0 ImagesCat. No.: HY-183808CAS No.: 1255918-84-3N-(1,2-Dithiolane-3-pentanoyl)-Glu-Ala is a derivative of DL-α-lipoic acid (HY-N0492). N-(1,2-Dithiolane-3-pentanoyl)-Glu-Ala can be used for the research of ischemic and ischemia-reperfusion injuries.
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(S)-Tsaokoin
0 ImagesCat. No.: HY-N14570CAS No.: 343605-41-4(S)-Tsaokoin is a natural terpenoid.
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Inositol phosphate amide-C5-NH2
0 ImagesCat. No.: HY-176883CAS No.: 889659-00-1Inositol phosphate amide-C5-NH2 (Compound 3) is inositol phosphate derivative.
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Roxibolone
0 ImagesCat. No.: HY-114835CAS No.: 60023-92-9Synonyms: BR-906Roxibolone (BR-906) is a 2-carboxy-1, 4-androstadien-3-one derivative. Roxibolone exerts potent anti-glucocorticoid activity and can counteract its catabolism. Roxibolone has no androgenic activity. Roxibolone can be used for research of glucocorticoid-related metabolic disorders.
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WAY-312491
0 ImagesWAY-312491 is an active molecule.
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5-Chloro DMT hydrochloride
0 Images5-chloro DMT (5-Chloro-N,N-dimethyltryptamine) hydrochloride is a Tryptamine (HY-B2132).
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cis-Vaccenic acid NHS ester
0 ImagesCat. No.: HY-185225CAS No.: 163069-97-4cis-Vaccenic acid NHS ester is an N-hydroxysuccinimide (NHS)-activated ester derivative of cis-vaccenic acid (HY-113427A) (C18:1 n-7), which is commonly used as a fatty acid labeling reagent or covalent modification reagent.
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6-(L-1,2,3-Trihydroxybutyl)-pterin
0 ImagesCat. No.: HY-W750595CAS No.: 13392-24-06-(L-1,2,3-Trihydroxybutyl)-pterin is a derivative of L-biopterin (HY-102015) and is the oxidized form of tetrahydro-L-biopterin (BH4) as well as D-biopterin. Co-ingestion of 6-(L-1,2,3-Trihydroxybutyl)-pterin (0.5%) with the carcinogen 4-dimethylaminoazobenzene reduces the incidence of 4-dimethylaminoazobenzene-induced liver tumors in rats. 6-(L-1,2,3-Trihydroxybutyl)-pterin has been used as an internal standard for the LC-MS quantification of biopterin and neopterin in rat plasma.
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Astaxanthin monopalmitate
0 ImagesCat. No.: HY-W750675CAS No.: 123159-02-4Synonyms: Astaxanthin palmitateAstaxanthin monopalmitate (Astaxanthin palmitate) is an esterified form of Astaxanthin (HY-B2163) (a carotenoid). Astaxanthin monopalmitate degradation resulted in a mixture of free and palmitate apo-astaxanthins. Carotenoids are important biological active, and may regulate cellular differentiation, growth control, photooxidative protection, cell membrane stability, photosynthesis, vision process and nutrition.
