1. Signaling Pathways
  2. Membrane Transporter/Ion Channel
    Neuronal Signaling
  3. GlyT
  4. GlyT Inhibitors

GlyT Inhibitors

GlyT1

GlyT2

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

GlyT Inhibitors & Antagonists
Product Name GlyT1 GlyT2 Purity
Bitopertin
GlyT1
  99.90%
Sarcosine
GlyT1
  98.0%
N-Arachidonylglycine  
GlyT2, IC50: 5.1 μM
99.45%
Stearoyl-L-carnitine chloride  
GlyT2
99.90%
RPI-GLYT2-82  
GlyT2, IC50: 544 nM
Org 24461
GLT1
 
Iclepertin
GLT1, IC50: 5.2 mM (In rat primary neurons )
GLT1, IC50: 5 nM (In human SK-N-MC cells)
  99.97%
Sarcosine-d3
GlyT1
  99.05%
Opiranserin hydrochloride  
GlyT2, IC50: 0.86 μM
99.62%
Stearoyl-L-carnitine-d3 chloride  
GlyT2
99.80%
PF-03463275
GlyT1
  98.79%
GlyT1 Inhibitor 1
rGlyT1, IC50: 38 nM
  98.59%
SSR504734
hGlyT1, IC50: 18 nM
rGlyT1, IC50: 15 nM
  99.42%
LY2365109 hydrochloride
hGlyT1, IC50: 15.8 nM nM
  98.69%
(Rac)-ALX 5407
hGlyT1, IC50: 2.8 nM
rGlyT1, IC50: 9.8 nM
 
ALX-1393  
GlyT2
≥99.0%
Sarcosine-15N
GlyT1
  99.92%
Tilapertin
GlyT1
 
TASP0315003
GlyT1
 
PF-03463275 hydrochloride
GLT1, Ki: 116 nM
 
Opiranserin  
GlyT2, IC50: 0.86 μM
GSK494581A
rGlyT1
 
Org 25935
GlyT1, IC50: 100 nM