1. Signaling Pathways
  2. Immunology/Inflammation
  3. IRAK
  4. IRAK Inhibitors

IRAK Inhibitors

IRAK1

IRAK4

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

IRAK Degraders & Inhibitors
Product Name IRAK1 IRAK4 Purity
Zimlovisertib  
IRAK4, IC50: 0.2 nM
99.84%
Emavusertib  
IRAK4, IC50: 57 nM
99.96%
Ginsenoside Rb1
IRAK-1
  98.75%
JH-X-119-01 hydrochloride
IRAK1
  98.15%
KT-474  
IRAK4
99.27%
Emavusertib hydrochloride  
IRAK4, IC50: 57 nM
KME-2780
IRAK1
IRAK4
HS-276
IRAK1, IC50: 264 nM
IRAK4, IC50: 2500 nM
98.59%
Zabedosertib  
IRAK4, IC50: 3.55 nM
99.12%
JH-X-119-01
IRAK-1, IC50: 9 nM
  ≥98.0%
PROTAC IRAK4 degrader-1  
IRAK4
99.72%
AZ1495
IRAK1, IC50: 23 nM
IRAK4, IC50: 5 nM
98.18%
HS-243
IRAK-1, IC50: 24 nM
IRAK4, IC50: 20 nM
99.88%
JNJ-1013
IRAK1, IC50: 72 nM
IRAK4, IC50: 443 nM
99.80%
IRAK4-IN-7  
IRAK4
99.36%
PF-06426779  
IRAK4, IC50: 0.3 nM
99.83%
GLPG2534
IRAK1, IC50: 179 nM
hIRAK4, IC50: 6.4 nM
mIRAK4, IC50: 3.5 nM
98.05%
IRAK-4 protein kinase inhibitor 2  
IRAK4, IC50: 4 μM
98.01%
PROTAC IRAK4 degrader-3  
IRAK4
Larotinib mesylate hydrate
IRAK-1, IC50: 167 nM
  98.66%
IRAK inhibitor 4 (trans)  
IRAK4
99.02%
HS271  
IRAK4, IC50: 7.2 μM
99.92%
IRAK4-IN-14  
IRAK4, IC50: 0.003 μM
Larotinib
IRAK1, IC50: 167 nM
 
IRAK4-IN-8  
IRAK4
IRAK4-IN-18  
IRAK4, IC50: 15 nM
PROTAC IRAK4 degrader-5  
IRAK4
IRAK4-IN-16  
IRAK4, IC50: 2.5 ± 0.8 nM
IRAK4-IN-9  
IRAK4, IC50: 1.5 nM
IRAK4-IN-10  
IRAK4, IC50: 1.5 nM
IRAK4-IN-13  
IRAK4, IC50: 0.6 nM
KTX-612  
IRAK4, DC50: 7 nM
PROTAC IRAK4 degrader-4  
IRAK4
BIO-7488  
hIRAK4, IC50: 0.6 nM
IRAK4-IN-20  
IRAK4, IC50: 3.55 nM
Ginsenoside Rb1 (Standard)
IRAK-1
 
KTX-497  
IRAK4, DC50: 3 nM
KTX-955  
IRAK4, IC50: 5 nM
IRAK4-IN-15  
IRAK4, IC50: 0.002 μM
IRAK4-IN-12  
IRAK4, IC50: 0.015 μM
IRAK4-IN-17  
IRAK4, IC50: 1.3 nM
PROTAC IRAK4 degrader-6  
IRAK4
IRAK4-IN-11  
IRAK4, IC50: .008 μM
IRAK4-IN-19  
IRAK4, IC50: 4.3 nM
HG-12-6  
IRAK4, IC50: 165 nM (Unphosphorylated inactive IRAK4 )
IRAK4, IC50: 2876 nM (Phosphorylated active IRAK4 )
GNE-2256  
IRAK4, Ki: 1.4 nM
IRAK4-IN-24  
IRAK4
IRAK4-IN-27  
IRAK4, IC50: 8.7 nM
PROTAC IRAK4 degrader-2  
IRAK4