1. Signaling Pathways
  2. MAPK/ERK Pathway
  3. JNK
  4. JNK Inhibitors

JNK Inhibitors

JNK1

JNK2

JNK3

JNK

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JNK Inhibitors, Activators, Modulators, Degraders & Ligands
Product Name JNK1 JNK2 JNK3 JNK Purity
SP600125
JNK1, IC50: 40 nM
JNK2, IC50: 40 nM
JNK3, IC50: 90 nM
  99.55%
Anisomycin      
JNK
99.82%
JNK-IN-8
JNK1, IC50: 4.7 nM
JNK2, IC50: 18.7 nM
JNK3, IC50: 1 nM
  99.67%
Astragaloside IV      
JNK
99.93%
Chloramphenicol      
JNK
99.96%
JNK1 ligand-1-NH-Ph-COOH
JNK1
      98.08%
Anti-inflammatory agent 99      
JNK
Gamma-glutamylcysteine
JNK1
      98.53%
Guggulsterone      
JNK
99.83%
Isovitexin
JNK1
JNK2
    99.90%
Ginsenoside Re      
JNK
99.92%
Tomatidine      
JNK
98.0%
JNK Inhibitor VIII
JNK1, Ki: 2 nM
JNK1, IC50: 45 nM
JNK2, Ki: 4 nM
JNK2, IC50: 160 nM
JNK3, Ki: 52 nM
  99.58%
Tanzisertib
JNK1, IC50: 61 nM
JNK2, IC50: 7 nM
JNK3, IC50: 6 nM
  99.98%
Bentamapimod
JNK1, IC50: 80 nM
JNK2, IC50: 90 nM
JNK3, IC50: 230 nM
  99.23%
D-JNKI-1      
JNK
99.29%
JNK-IN-7
JNK1, IC50: 1.5 nM
JNK2, IC50: 2 nM
JNK3, IC50: 0.7 nM
  98.17%
CC-90001
JNK1
JNK2
    99.98%
CC-401 hydrochloride      
JNK, Ki: 25-50 nM
99.35%
TNG348
JNK1
      99.74%
AS601245
hJNK1, IC50: 150 nM
hJNK2, IC50: 220 nM
hJNK3, IC50: 70 nM
  98.19%
BI-78D3      
JNK, IC50: 280 nM
99.85%
Tomatidine hydrochloride      
JNK
99.70%
Seratrodast      
JNK
99.59%
Geranial
JNK2
 
JNK3
  99.51%
Kanamycins sulfate
JNK1
      99.22%
Prostaglandin A2
JNK1
      99.9%
Cornuside
JNK1
JNK2
    99.99%
TCS JNK 5a  
JNK2, pIC50: 6.5
JNK3, pIC50: 6.7
  99.40%
DB07268
JNK1, IC50: 9 nM
      99.04%
Juglanin      
JNK
99.76%
Loureirin B      
JNK
99.96%
Daphnoretin      
JNK
99.83%
Indirubin-3′-oxime
JNK1, IC50: 0.8 μM
JNK2, IC50: 1.4 μM
JNK3, IC50: 1 μM
  99.10%
PT109
JNK1, IC50: 0.143 μM
JNK2, IC50: 0.831 μM
JNK3, IC50: 0.285 μM
  99.20%
Armepavine      
JNK
99.53%
CC-401      
JNK, Ki: 25-50 nM
99.63%
JNK3 inhibitor-4
JNK1, IC50: 143.9 nM
JNK2, IC50: 298.2 nM
JNK3, IC50: 1.0 nM
  99.37%
Viridicatol      
JNK
99.93%
SR-3576    
JNK3, IC50: 7 nM
  99.75%
Ombuoside
JNK1
      99.68%
J30-8    
JNK3, IC50: 40 nM
  99.51%
SR-3306      
JNK
99.0%
IQ-1S free acid
JNK1, Kd: 240 nM
JNK2, Kd: 360 nM
JNK3, Kd: 100 nM
  99.28%
CEP-1347
JNK1
      98.50%
Sugiol
JNK1
JNK2
    99.88%
MPT0B392      
JNK
99.63%
Vitexin-4''-O-glucoside      
JNK
99.86%
L-JNKI-1      
JNK
99.01%
JTP10-△-TATi TFA
JNK1, IC50: 1.16 μM
JNK2, IC50: 92 nM
JNK3, IC50: 1.2 μM
  99.65%
SX 011
JNK1, IC50: > 300,000 nM
JNK2, IC50: 100 nM
    99.33%
Wnt/β-catenin-IN-6      
JNK
98.34%
IQ-3
JNK1, Kd: 0.24 μM
JNK2, Kd: 0.29 μM
JNK3, Kd: 0.066 μM
  99.38%
JNK-1-IN-5
JNK1
      99.63%
15(R)-Lipoxin A4
JNK1
JNK2
JNK3
  98.3%
JNK-IN-11
JNK1, IC50: 1.8 μM
JNK2, IC50: 21.4 μM
JNK3, IC50: 2.2 μM
  98.01%
JNK-IN-13  
JNK2, IC50: 500 nM
JNK3, IC50: 290 nM
 
JNK-9L
JNK1, IC50: 0.099 μM
 
JNK3, IC50: 0.148 μM
  98.06%
Salicortin      
JNK
JTP10-△-R9 TFA
JNK1, IC50: 1.1 μM
JNK2, IC50: 89 nM
JNK3, IC50: 1.2 μM
  99.95%
JNK-IN-16      
JNK, IC50: 72 nM
99.82%
YL5084
JNK1, IC50: 2173 nM
JNK2, IC50: 70 nM
JNK3, IC50: 84 nM
 
JNK-IN-14
JNK1, IC50: 1.82 nM
JNK2, IC50: 10.5 nM
JNK3, IC50: 10.5 nM
 
(-)-Zuonin A
JNK1, IC50: 1.7 μM
JNK2, IC50: 2.9 μM
JNK3, IC50: 1.74 μM
  99.99%
IQ-1S
JNK1, Kd: 390 nM
JNK2, Kd: 360 nM
JNK3, Kd: 87 nM
 
JNK-1-IN-1
JNK1
     
JNK1 degrader-1
JNK1
     
Cm-CATH2      
JNK
JNK-IN-25
JNK1, IC50: 1.54 nM
JNK2, IC50: 1.99 nM
JNK3, IC50: 0.75 nM
 
Aloisine A      
JNK, IC50: 3-10 μM
JAK3-IN-13
JNK1, IC50: 4728 nM
JNK2, IC50: 2039 nM
JNK3, IC50: 8 nM
 
GSK3-IN-10    
JNK3, IC50: 2900 nM
 
JNK2/MKK7 PPI-IN-1  
JNK2, IC50: 0.99 μM
JNK2, Kd: 81.6 μM
   
Ginsenoside Re (Standard)      
JNK
JNK3 inhibitor-7
JNK1, IC50: 1039 nM
JNK2, IC50: 973 nM
JNK3, IC50: 53 nM
 
JNK3-IN-11    
JNK3, IC50: 2.08 nM
 
Lucidone      
JNK
ERK2 IN-5    
JNK3, Ki: 550 nM
 
Cernuumolide J    
JNK3
 
JNK3/Wnt/β-catenin modulator-1    
JNK3
 
JNK3 inhibitor-5
JNK1, IC50: 82.7 nM
JNK2, IC50: 29.4 nM
JNK3, IC50: 0.379 nM
 
Necrostatin-21    
JNK3
 
JNK3 inhibitor-8
JNK1, IC50: >10000 nM
JNK2, IC50: 2203 nM
JNK3, IC50: 21 nM
 
PROTAC JNK1-targeted-1
JNK1, DC50: 10 nM
     
MR2938      
JNK
JNK3 inhibitor-3
JNK1, IC50: 147.8 nM
JNK2, IC50: 44 nM
JNK3, IC50: 4.1 nM
 
JNK1 ligand-1
JNK1
     
SP600125 (GMP)
JNK1, IC50: 40 nM
JNK2, IC50: 40 nM
JNK3, IC50: 90 nM
 
JNK2/3-IN-1  
JNK2
JNK3
 
JNK3-IN-10    
hJNK3, IC50: 0.257 nM
 
Hydrostatin-TL1      
JNK
JNK-1-IN-4
JNK1, IC50: 2.7 nM
JNK2, IC50: 19.0 nM
JNK3, IC50: 9.0 nM
 
TOPK-p38/JNK-IN-1      
JNK
ZG-10
JNK1, IC50: 809 nM
JNK2, IC50: 1140 nM
JNK3, IC50: 709 nM
 
JNK3 inhibitor-9    
JNK3, IC50: 12 nM
 
Ophiopogonin B      
JNK
99.90%
Cyy-272
JNK1, IC50: 1.25 μM
JNK2, IC50: 1.07 μM
JNK3, IC50: 1.24 μM
 
JNK3 inhibitor-2
JNK1, IC50: >100 μM
JNK2, IC50: >100 μM
JNK3, IC50: 0.25 μM
 
(3S)-Tanzisertib hydrochloride
JNK1, IC50: 61 nM
JNK2, IC50: 7 nM
JNK3, IC50: 6 nM