1. Signaling Pathways
  2. Cell Cycle/DNA Damage
    Metabolic Enzyme/Protease
    Vitamin D Related/Nuclear Receptor
  3. PPAR
  4. PPAR Inhibitors

PPAR Inhibitors

PPARα

PPARβ/δ

PPARγ

PPAR

PPARδ

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

PPAR Inhibitors, Agonists, Antagonists, Activators, Modulators, Inducers & Ligands
Product Name PPARα PPARβ/δ PPARγ PPAR PPARδ Purity
Retinoic acid
PPARα, Kd: 103 nM
PPARα, IC50: 14 nM
PPARβ/δ, Kd: 17 nM
RARβ, IC50: 14 nM
PPARγ, Kd: 178 nM
PPARγ, IC50: 14 nM
    99.81%
Rosiglitazone    
PPARγ, Kd: 40 nM
PPARγ, EC50: 60 nM
    99.94%
GW9662
PPARα, IC50: 32 nM
PPARδ, IC50: 2000 nM
PPARγ, IC50: 3.3 nM
    99.98%
5-Aminosalicylic Acid    
PPARγ
    99.97%
Fenofibrate
PPARα, IC50: 30 μM
        99.97%
AM9053
PPARα
        98.36%
NO-Pravastatin
PPARα
 
PPARγ
   
MRL20    
PPAR-γ, EC50: 10 nM
   
GW6471
PPARα
        99.64%
Pioglitazone
hPPARα, EC50: 100 μM
mouse PPARα, EC50: 100 μM
hPPARδ, EC50: 43 μM
hPPARγ, EC50: 0.93 μM
mouse PPARγ, EC50: 0.99 μM
    99.70%
Pirinixic acid
PPARα, EC50: 0.63 μM
 
PPARγ, EC50: 32 μM
    99.34%
Troglitazone    
PPARγ, EC50: 550 nM (Human PPARγ)
    99.78%
Icariin
PPARα
        99.06%
T0070907
PPARα, Ki: 0.85 μM
PPARδ, Ki: 1.8 μM
PPARγ, Ki: 1 nM
    99.98%
GW7647
PPARα, EC50: 6 nM (Human PPARα)
PPARδ, EC50: 6.2 μM (Human PPARδ)
PPARγ, EC50: 1.1 μM (Human PPARγ)
    99.45%
Daidzein
PPAR-α
 
PPAR-γ
    99.81%
Astaxanthin    
PPARγ
    98.0%
Sodium propionate    
PPAR-γ
    99.0%
Oleuropein    
PPARγ
    99.97%
GW 501516  
PPARδ, EC50: 1.1 nM
      99.27%
Anandamide      
PPAR
  ≥99.0%
Elafibranor
PPAR-α, EC50: 45 nM
PPAR-δ, EC50: 175 nM
      99.66%
Pemafibrate
h-PPARα, EC50: 1 nM
PPARδ, EC50: 1.58 μM
h-PPARγ, EC50: 1.1 μM
    99.85%
Magnolol    
PPARγ, EC50: 17.7 μM
    99.84%
Fucoxanthin
PPARα
 
PPARγ
    99.38%
Pioglitazone hydrochloride
PPARα, EC50: 0.93 μM (Human PPARα)
PPARδ, EC50: 0.01 μM (Human PPARδ)
PPARγ, EC50: 43 μM (Human PPARγ)
    99.97%
Retinoic acid (Standard)
PPARα
PPARβ/δ
RARβ
PPARγ
   
Glabridin    
PPARγ, EC50: 6.1 μM
    99.98%
Bezafibrate
hPPARα, EC50: 50 μM
hPPARδ, EC50: 20 μM
hPPARγ, EC50: 60 μM
    99.83%
Oleoylethanolamide
PPAR-α
        98.19%
Inclisiran sodium    
PPARγ
    99.08%
GSK3787  
PPARδ, pIC50: 6.6 nM
      99.94%
GW1929    
PPAR-γ, pEC50: 8.56 (Human PPAR-γ)
    99.93%
GW0742
PPARα, EC50: 1.1 μM
PPARδ, EC50: 1 nM
PPARγ, EC50: 2 μM
    99.64%
Inclisiran    
PPARγ
    99.48%
Palacaparib      
PPAR
  98.30%
Dehydroepiandrosterone sulfate
PPARα
        99.93%
Rosiglitazone maleate    
PPARγ1, EC50: 30 nM
PPARγ2, EC50: 100 nM
    99.73%
Seladelpar
PPAR-α, EC50: 1600 nM
PPAR-δ, EC50: 2 nM
      99.75%
Fmoc-leucine    
PPARγ
    99.91%
CDDO-Im
PPARα, Ki: 232 nM
 
PPARγ, Ki: 344 nM
    99.30%
9''-Methyl salvianolate B    
PPARγ
    99.54%
GSK0660  
PPARβ/δ, IC50: 155 nM
      99.49%
FH535      
PPAR
  99.95%
1-Methyladenosine    
PPAR-γ
    99.92%
Candesartan    
PPAR-γ
    98.10%
Gemfibrozil
PPAR-α
        99.91%
Palmitelaidic acid
PPARα
        99.4%
Sodium acetate trihydrate, meets analytical specification of Ph. Eur. BP USP FCC E262, ≤0.00002% Al
PPARα
        99.7%
Dehydroepiandrosterone sulfate sodium
PPARα
        99.96%
1,2-DLPC
PPARα
        98.0%
Ginsenoside Rh1    
PPAR-γ
    98.72%
Hexadecanamide
PPARα
        99.64%
Chiglitazar
PPARα, EC50: 1.8 μM
PPARδ, EC50: 1.7 μM
PPARγ, EC50: 0.08 μM
    99.81%
Bilobetin
PPARα
        99.71%
Eupatilin
PPARα
        98.90%
Perfluoro(2-methyl-3-oxahexanoic) acid
PPARα, EC50: 2.1 μM
        99.41%
Clofibrate
PPARα, EC50: 50 μM
 
PPARγ, EC50: 500 μM
    99.61%
Alpinetin    
PPAR-γ
    99.51%
Rosiglitazone hydrochloride    
PPARγ, EC50: 60 nM
PPARγ, Kd: 40 nM
    99.81%
Bavachinin
PPARα, IC50: 21.043 μM
PPARδ, IC50: 12.819 μM
PPAR-γ, IC50: 0.622 μM
    99.95%
Saroglitazar
PPARα, EC50: 0.65 pM (HepG2 cell)
 
PPARγ, EC50: 3 nM (HepG2 cell)
    98.22%
Agrimol B    
PPARγ
    99.75%
Fenofibric acid
PPARα, EC50: 22.4 μM
PPARδ, EC50: 1.06 μM
PPARγ, EC50: 1.47 μM
    99.94%
Magnesium acetate tetrahydrate
PPARα
        99.47%
FX-909    
PPARγ
    99.79%
15-Deoxy-Δ-12,14-prostaglandin J2    
PPARγ, EC50: 2 μM
    ≥99.0%
Sinigrin    
PPARγ
    99.97%
15-keto-Prostaglandin E2    
PPARγ
    ≥99.0%
Ophiopogonin D
PPARα
        99.80%
D-Arabinose    
PPAR-γ
    ≥99.0%
Lobeglitazone
PPARα, EC50: 546.3 nM
 
PPARγ, EC50: 137.4 nM
   
MTX-531    
PPARγ, EC50: 3.4 μM
    99.87%
Urolithin D    
PPARγ
    99.72%
Perfluorobutanesulfonic acid    
PPARγ
    98.0%
γ-Glutamylvaline    
PPAR-γ
    99.94%
Avicularin    
PPARγ
    99.80%
Alisol A
PPARα
        99.59%
SR1664    
PPAR-γ, IC50: 80 nM
    98.12%
Gypenoside XLIX
PPAR-α
        99.88%
Daidzein (Standard)
PPAR-α
 
PPAR-γ
   
Seladelpar sodium  
PPAR-δ, EC50: 2 nM
      98.59%
AMG131    
PPARγ
    98.99%
NXT629
hPPARα, IC50: 77 nM
hPPARδ, IC50: 6 μM
hPPARγ, IC50: 15 μM
    98.75%
Phellopterin    
PPARγ
    99.94%
L-165041  
PPARδ, Ki: 6 nM
PPARγ, Ki: 730 nM
    99.12%
Ciprofibrate
PPARα
        99.93%
Glabrone    
PPAR-γ
    99.08%
SDPC    
PPARγ
    98.0%
Perfluorononanoic acid
PPARα
        99.9%
Clitorin
PPARα
        99.45%
DG172 dihydrochloride  
PPARβ/δ, IC50: 27 nM
      99.51%
Oroxin A    
PPARγ
    99.76%
Oroxylin A-7-O-glucuronide    
PPARγ
    99.83%
Rubrofusarin gentiobioside    
PPAR-γ
    99.04%
Leriglitazone    
PPAR-γ, EC50: 9 μM
    99.23%
(E)-Osmundacetone
PPARα
        99.81%
Raspberry ketone
PPAR-α
        99.95%
Norathyriol
PPARα, IC50: 92.8 μM
PPARβ, IC50: 102.4 μM
PPARγ, IC50: 153.5 μM
    99.74%
Azemiglitazone potassium    
PPAR-γ, IC50: 18.25 μM
    98.94%
F44-A13
PPARα
PPARβ
     
25-Hydroxytachysterol3    
PPARγ
    98.07%
Licarin B    
PPARγ
    99.93%
Balaglitazone    
PPARγ, EC50: 351 nM (Human PPARγ)
    99.25%
Saroglitazar magnesium
PPARα, EC50: 0.65 pM (HepG2 cell)
 
PPARγ, EC50: 3 nM (HepG2 cell)
    98.85%
Leriglitazone hydrochloride    
PPAR-γ, EC50: 9 μM
    99.64%
BAY-4931    
PPAR-γ, IC50: 0.17 nM (RT112-FABP4-NLucP cellular reporter assay)
mouse PPARγ, IC50: 0.14 nM (GAL4-NHR-LBD one hybrid reporter assay )
hPPARγ, IC50: 0.40 nM (GAL4-NHR-LBD one hybrid reporter assay )
    98.72%
PPARγ-IN-2    
PPARγ
    99.65%
Falcarindiol    
PPARγ
    99.48%
(10E,12Z)-Octadeca-10,12-dienoic acid
PPARα
        99.10%
PPARα/γ agonist 1
PPARα, EC50: 28 nM
 
PPARγ, EC50: 69 nM
    99.69%
FTX-6746    
PPARγ
    99.07%
GSK1820795A    
hPPARγ, EC50: 0.25 μM
mouse PPARγ, EC50: 0.27 μM
    99.80%
SR 16832    
PPARγ
    99.58%
Dehydroepiandrosterone sulfate sodium-d6
PPARα
        99.61%
Amezalpat
PPARα, IC50: 58 nM
        99.85%
Inolitazone dihydrochloride    
PPARγ
    98.45%
Darglitazone    
PPAR-γ
    99.19%
Drupanin
PPARα, EC50: 39.0 μM
 
PPARγ, EC50: 14.6 μM
    99.35%
Edaglitazone
PPARα, EC50: 1053 nM
 
PPARγ, EC50: 35.6 nM
    99.57%
Icariin (Standard)
PPARα
       
Ertiprotafib
PPARα, EC50: ~1 μM
PPARβ, EC50: ~1 μM
      98.13%
ST247  
PPARβ/δ
      99.88%
Mifobate    
PPARγ, IC50: 140 μM
    99.85%
HWL-088  
PPARδ, EC50: 570.9 nM
      98.61%
Indeglitazar
PPARα
PPARδ
PPARγ
    98.52%
Perfluoropentanoic acid    
PPARγ
 
PPARδ
98.0%
Psammaplin A    
PPARγ
   
H-​Trp-​Glu-​OH    
PPARγ, Kd: 8 μM
    99.95%
4-O-Methyl honokiol    
PPARγ
    98.76%
Cefminox sodium    
PPARγ
    99.83%
Garcinia cambogia extract    
PPARγ2
   
CUDA
PPARα
        99.83%
1,1'-(Azodicarbonyl)-dipiperidine
PPARα
 
PPAR-γ
 
PPARδ
≥98.0%
Netoglitazone    
PPARγ
    99.92%
Angeloylgomisin H    
PPAR-γ
    99.79%
GW 9578
mouse PPARα, EC50: 5 nM
h-PPARα, EC50: 50 nM
        99.6%
BMS-687453
PPARα, IC50: 260 nM (Human PPARα)
        99.31%
Fenofibric acid (Standard)
PPARα
PPARδ
PPARγ
   
Tartronic acid    
PPARγ
    ≥98.0%
6-​Thioinosine    
PPAR-γ
    99.31%
FK614    
PPAR-γ
    99.97%
Alisol A 24-acetate
PPARα
 
PPAR-γ
    98.0%
1-O-Hexadecylglycerol    
PPAR-γ
    99.96%
Etrinabdione    
PPARγ
    99.16%
MRL-24    
PPARγ
    99.58%
Cichoriin    
PPAR-γ
    99.9%
Gemfibrozil (Standard)
PPAR-α
       
Sulindac sulfone    
PPARγ
    98.10%
ZLY06    
PPARγ, IC50: 237 nM
 
PPARδ, IC50: 341 nM
98.75%
Fenofibrate (Standard)
PPARα
       
Glabridin (Standard)    
PPARγ
   
Aleglitazar
PPARα, IC50: 38 nM
 
PPARγ, IC50: 19 nM
    99.74%
Dehydroepiandrosterone sulfate (Standard)
PPARα
       
Lobeglitazone sulfate
PPARα, EC50: 546.3 nM
 
PPARγ, EC50: 137.4 nM
    99.63%
Adelmidrol    
PPARγ
    98.0%
10-Nitrolinoleic acid    
PPARγ, IC50: 0.22 μM
   
CP-868388 free base
hPPARα, Ki: 10.8 nM
 
hPPARγ, Ki: 3.47 μM
    99.66%
LT175
hPPARα, EC50: 0.22 μM
mPPARα, EC50: 0.26 μM
 
hPPARγ, EC50: 0.48 μM
    99.46%
PPARα/δ agonist 1
PPARα, EC50: 7 nM
 
PPARγ, EC50: 1316.1 nM
 
PPARδ, EC50: 8.4 nM
99.59%
PPAR agonist 5
PPARα, EC50: 3.20 μM
PPARβ/δ, EC50: 1.51 μM
PPARγ, EC50: 1.92 μM
   
Methyl oleanonate    
PPARγ
    99.81%
(±)4-HDHA    
PPARγ
    99.05%
SR 11023    
PPARγ, IC50: 108 nM
    99.55%
9(10)-Nitrooleate
PPARα
PPARβ/δ
PPARγ
    99.0%
Dehydroepiandrosterone sulfate-d6 sodium dihydrate
PPARα
        99.9%
YS121
PPAR-α, EC50: 1 μM
 
PPAR-γ, EC50: 3.6 μM
    99.74%
BAY-0069    
hPPARγ, IC50: 6.3 nM
mouse PPARγ, IC50: 24 nM
    98.07%
Clofibrate (Standard)
PPARα
 
PPARγ
   
Vitisin A    
PPAR-γ
   
PPARγ agonist 14    
PPARγ, EC50: 2.4 μM
    98.0%
Rivoglitazone    
PPARγ, EC50: 0.22 μM
    98.59%
PPARγ phosphorylation inhibitor 1    
PPARγ, IC50: 24 nM
    99.81%
Saringosterol    
PPARγ
   
PPARα agonist 6
PPARα
        99.79%
BGT-002
PPARα
        99.35%
BAY-5094    
PPAR-γ
    98.04%
MA-0204  
PPARδ, EC50: 0.4 nM (in human)
PPARδ, EC50: 7.9 nM (in mouse)
PPARδ, EC50: 10 nM (in rat)
      99.31%
Eupatilin (Standard)
PPARα
       
Sinigrin hydrate    
PPARγ
    99.92%
13-Oxo-9E,11E-octadecadienoic acid
PPARα
       
GSK376501A    
PPARγ
    99.06%
Perfluorotetradecanoic acid    
hPPARγ, Kd: 157.8 μM
    98.0%
PPAR agonist 1
PPARα
 
PPARγ
    98.39%
E0924G  
PPARδ, EC50: 2.82 μM
      99.17%
SKLB102    
PPAR-γ
    98.0%
Chiglitazar sodium
PPARα, EC50: 1.8 μM
PPAR-δ, EC50: 1.7 μM
PPAR-γ, EC50: 0.08 μM
    98.33%
Tibric acid
PPARα
       
9(S)-HOTrE
PPARα
        99.9%
Arhalofenate    
PPAR-γ
    99.85%
PPARα agonist 2
PPARα, EC50: 37 nM
        98.9%
Rosiglitazone potassium    
PPARγ, Kd: 40 nM
PPARγ, EC50: 60 nM
    99.13%
Pparδ agonist 5        
PPARδ, EC50: 0.335 μM
ABP/PPAR modulator 1
PPARα, EC50: 9.19 μM
 
PPARγ, EC50: 2.20 μM
 
PPARδ, EC50: 1.58 μM
Seladelpar (lysine dihydrate)        
PPARδ, EC50: 2 nM
99.51%
Pioglitazone potassium
hPPARα, EC50: 100 μM
mouse PPARα, EC50: 100 μM
hPPARδ, EC50: 43 μM
mouse PPARγ, EC50: 0.99 μM
h-PPARγ, EC50: 0.93 μM
   
GED 0507-34-Levo    
PPARγ
   
Inolitazone hydrochloride hydrate    
PPARγ
   
PPARα/δ agonist 2
PPARα, EC50: 3255 nM
PPARβ/δ, EC50: 1475 nM
     
Ciprofibrate impurity A
PPARα
       
BMS711939
hPPARα, IC50: 4 nM
 
hPPARγ, IC50: 4.5 μM
   
MBX-102 acid    
PPARγ
   
Tibesaikosaponin V    
PPARγ
   
PPARγ-IN-3    
PPARγ
   
PPARγ agonist-23    
PPARγ, EC50: 0.32 μM
   
Esculeogenin A
PPARα
       
EL244    
PPAR-γ, IC50: 1.3 μM
    99.55%
PPAR agonist 4
PPARα, EC50: 0.7 μM
 
PPARγ, EC50: 1.8 μM
 
PPARδ, EC50: 0.7 μM
PPARγ modulator-4    
PPARγ, Kd: 3.75 μM
   
LJ570
PPARα, EC50: 1.05 μM
 
PPARγ, EC50: 0.12 μM
   
PPARγ/δ modulator 2    
PPARγ
 
PPARδ
Caulophyllogenin    
PPARγ, EC50: 12.6 μM
   
PA-082    
PPAR-γ
   
PPAR agonist 8
PPARα, Kd: 0.576 μM
 
PPARγ, Kd: 2.06 μM
 
PPARδ, Kd: 1.45 μM
Pparδ agonist 1  
PPARδ, EC50: 5.06 nM
     
Neoambrosin    
PPARγ
   
Darglitazone Sodium    
PPAR-γ
   
Rac-Pemafibrate
h-PPARα, EC50: 1 nM
h-PPARδ, EC50: 1.7 μM
     
PPARγ/δ modulator 1    
PPARγ, Ki: 5.31 μM
 
PPARδ, Ki: 14.4 nM
ESP-31015
PPARα
       
Imiglitazar
PPARα, EC50: 67 nM
 
PPARγ1, EC50: 31 nM
   
GW1929 hydrochloride    
hPPARγ, pKi: 8.84
   
Fonadelpar  
PPARδ
     
GSK 1997132B    
PPAR-γ, pEC50: 8
   
AZD4619
PPARα
       
XYQ3-B11
PPARα, EC50: 8.33 μM
       
AI 3-25755    
PPAR-γ
   
Cinoxate    
PPARγ, Ki: 18 μM
   
HD202A    
PPARγ1
   
Cevoglitazar
PPARα
 
PPARγ
   
Pparδ agonist 2  
PPARδ
     
HSD17B13/PPAR modulator-1
PPARα, EC50: 1.55 μM
 
PPARγ, EC50: 0.01 μM
 
PPARδ, EC50: 0.12 μM
PPARγ agonist 16    
PPAR-γ, IC50: 1790 nM
   
Apo-12'-lycopenal    
PPAR-γ
   
KD-3010  
PPARδ
     
PPARα/δ agonist 4
PPARα, EC50: 0.36 nM
 
PPARγ, EC50: 160.84 nM
 
PPARδ, EC50: 1.31 nM
PPARγ agonist 8    
PPARγ
   
DS-6930    
PPARγ, EC50: 41 nM
   
Romazarit
PPARα
       
(E)-Osmundacetone (Standard)
PPARα
       
GW-9820
PPARα, EC50: 0.37 μM
 
PPARγ, EC50: 0.288 μM
   
Ginsenoside Rh1 (Standard)    
PPAR-γ
   
15-Deoxy-Δ12,14-Prostaglandin J2-2-glyceryl ester    
PPARγ, EC50: 2 μM
   
PPARα agonist 5
PPARα, EC50: 3 nM
 
PPAR-γ, EC50: 1.66 μM
 
PPARδ, EC50: >25 μM
KRP-105
PPARα
       
S-Petasin    
PPARγ
   
SR2595    
PPARγ, IC50: 30 nM
   
Zaltoprofen sulfoxide    
PPAR-γ
   
LTD4 antagonist 3    
PPAR-γ
   
PPARδ agonist 10        
PPARδ, EC50: 0.053 μM (hPPARδ)
PPARδ, EC50: 0.30 μM (mPPARδ)
PPARγ modulator-1    
PPAR-γ
   
L-783483        
PPARδ
DN203316
hPPARα, EC50: 8 μM
hPPARδ, EC50: 0.02 μM
h-PPARγ, EC50: >10 μM
   
PPARγ agonist 19    
PPARγ
   
PPARγ agonist 2    
PPARγ
   
PPARα/δ agonist 3
PPARα, IC50: 5.6 nM
 
PPARγ, IC50: 1278 nM
 
PPARδ, IC50: 3.4 nM
PPARγ agonist-22    
PPAR-γ
   
CAY10410    
PPARγ
   
LCI765    
PPARγ, EC50: 0.07 nM
   
Hydrangeic acid    
PPARγ2
   
Mesalamine impurity P      
PPAR
 
PPARγ agonist-21    
PPAR-γ, EC50: 3.12 μM
   
15-LOX-IN-2    
PPARγ
   
Dehydroepiandrosterone sulfate sodium (Standard)
PPARα
       
GW7845    
PPARγ
   
(E/Z)-Oleamide
mouse PPARα
        99.97%
DN-108    
PPARγ
   
FSVVPSPK    
PPARγ
   
PPARα agonist 1
hPPARα
       
Ciprofibrate (Standard)
PPARα
       
4,5-DiHDPA lactone    
PPARγ
   
PPARγ modulator-3    
PPARγ, Kd: 186 nM
   
PPARγ-IN-5    
PPARγ
   
YGT-31    
PPARγ, IC50: 1.72 μM
PPARγ, Ki: 0.62 μM
   
PPARγ/GR modulator 1    
PPARγ, Ki: 3.3 μM
   
Avicularin (Standard)    
PPARγ
   
Porphyra 334    
PPARγ2
   
PPARα/γ agonist 2
PPARα, EC50: 0.95 μM
 
PPARγ, EC50: 0.91 μM
   
PPARδ agonist 13
PPARα, EC50: >10000 nM
 
PPARγ, EC50: >10000 nM
 
PPARδ, EC50: 0.5 nM
PPARα/γ agonist 4
PPARα
 
PPAR-γ
   
PPARγ modulator-2    
PPARγ, IC50: 41 nM
   
PPARα/δ antagonist-1
PPARα, IC50: 0.113 μM
     
PPARδ, IC50: 0.025 μM
DSO-5a    
PPARγ
   
sEH/PPARδ modulator 1        
PPARδ, EC50: 0.12 μM
CF-Vanillin
PPARα
       
Elaidyl-sulfamide
PPARα
       
Rosiglitazone sodium    
PPARγ1, EC50: 30 nM
PPARγ2, EC50: 100 nM
   
Prostaglandin A3    
PPAR-γ, Ki: 188 μM
   
PT-S58  
PPARβ/δ, IC50: 98 nM
     
CC618  
PPARδ, IC50: 10 μM
      99.94%
Prostaglandin B3    
PPARγ
   
Sitofibrate
PPAR-α
       
T2384    
PPARγ
   
SR-1903    
PPARγ, IC50: 209 nM
   
Inolitazone    
PPARγ
   
17-Oxo-7(Z),10(Z),13(Z),15(E),19(Z)-docosapentaenoic acid    
PPARγ
   
GW 2433
PPARα
     
PPARδ
ZINC17167211
PPAR-α, EC50: 0.16 nM
       
TZD18
hPPARα, IC50: 0.028 μM
 
hPPARγ, IC50: 0.057 μM
 
PPARδ, IC50: >10 μM
AVE-8134
PPARα, EC50: 100 nM (Human PPARα)
       
GW409544
PPARα, EC50: 2.3 nM
 
PPAR-γ, EC50: 0.28 nM
   
CLX-0921    
PPARγ, IC50: 1.54 μM
   
N-Octadecyl-N'-propyl-sulfamide
PPARα
       
NS-220
PPARα, EC50: 19 nM
 
PPARγ, EC50: 9.6 μM
 
PPARδ, EC50: >1 mM
Alisol A (Standard)
PPARα
       
PPARα-MO-1
PPARα