1. Signaling Pathways
  2. Cell Cycle/DNA Damage
  3. NEKs
  4. NEKs Inhibitors

NEKs Inhibitors

NEK1

NEK2

NEK4

NEK6

NEK7

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Sorry. There is currently no product that acts on isoform together.

Please try each isoform separately.

NEKs Inhibitors & Degraders
Product Name NEK1 NEK2 NEK4 NEK6 NEK7 Purity
LC-04-045        
NEK7, DC50: 7 nM
99.56%
Ofirnoflastum        
NEK7, IC50: 46 nM
99.93%
T-1101 tosylate  
NEK2
      98.91%
BSc5367
NEK1, IC50: 11.5 nM
        98.21%
NEK7 degrader-3        
NEK7, DC50: 33.1 nM
CG-1521  
NEK2
     
AP4-43    
NEK4
   
NK7-902 diTFA        
NEK7
99.88%
MBM-55  
NEK2, IC50: 1 nM
      99.94%
INH1  
NEK2
      99.85%
INH154  
NEK2
      99.89%
MRT-3486        
NEK7
99.62%
ZINC05007751      
NEK6, IC50: 3.4 μM
  99.33%
JH295  
NEK2, IC50: 770 nM
      98.66%
NBI-961  
NEK2
      99.73%
SLC3037        
NEK7
99.85%
NEK7 degrader-1        
NEK7, DC50: 9 nM
99.94%
INH6  
NEK2
      99.53%
TAI-1  
NEK2
      98.60%
CK7
NEK1
        99.72%
NLRP3-IN-79        
NEK7
99.10%
ABS-752 hydrochloride        
NEK7
98.81%
MBM-17S  
NEK2, IC50: 3 nM
     
JH295 hydrate  
NEK2, IC50: 770 nM
      99.0%
Nek2/Hec1-IN-2  
NEK2
      98.0%
Nek2-IN-4  
NEK2, IC50: 15 nM
     
MBM-55S  
NEK2, IC50: 1 nM
     
MBM-17  
NEK2, IC50: 3 nM
     
T-1101  
NEK2
     
NEK7 degrader-4        
NEK7, DC50: 9 nM
Nek2-IN-6  
NEK2
     
GSK461364 analogue 1  
NEK2, IC50: 21 nM
     
NEK7 degrader-2        
NEK7
PPARγ agonist-21        
NEK7
Nek2-IN-5  
NEK2
      99.17%