2. Signaling Pathways
  3. GPCR/G Protein
  4. PACAP Receptor
  5. PAC1 Receptor Isoform
  6. PAC1 Receptor Antagonist

PAC1 Receptor Antagonist

PAC1 Receptor Antagonist (1):

Cat. No. Product Name Effect Purity
  • HY-147557
    PA-915
    		Antagonist 99.17%
    PA-915 (PAC1R antagonist 1) is a potent and orally active antagonist of PAC1 receptor. PA-915 inhibits pituitary adenylate cyclase-activating polypeptide (PACAP)-induced CREB phosphorylation. PA-915 can inhibit PACAP- and nerve injury-induced allodynia. PA-915 can be used for the research of neuropathic pain.