CP-464709
CP-464709 is a Ghrelin receptor agonist that can penetrate the blood-brain barrier. CP-464709 causes an increase in blood pressure by activating pre sympathetic neurons in the spinal cord. CP-464709 causes biphasic blood pressure response when administered intravenously, while intrathecal administration only causes pressor. CP-464709 can be used for research on cardiovascular conditions.
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- CAS No.: 193272-70-7
- Formule: C28H31F5N6O4
- Masse moléculaire:610.58
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
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Activité biologique
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Chemical Information
- Pureté et documentation
- Références
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Help & FAQs
Activité biologique
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Cell Line
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Type | Value | Description | References |
|---|---|---|---|---|
| Pituitary gland cell | EC50 |
3 nM
Compound: 4, (CP-464709-18)
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In vitro effective concentration required for 50% stimulation of GH release in rat pituitary cell cultures.
In vitro effective concentration required for 50% stimulation of GH release in rat pituitary cell cultures.
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[PMID: 12392732] |
Chemical Information
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CAS No. 193272-70-7
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Masse moléculaire 610.58
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Formule C28H31F5N6O4
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SMILES
CC(C)(N)C(N[C@H](COCC1=CC=C(F)C=C1F)C(N(C[C@]23CC4=NC=CC=C4)CCC2=NN(CC(F)(F)F)C3=O)=O)=O
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
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