PDE5-IN-15
PDE5-IN-15 (compound 21) is a xanthine derivative and PDE5 inhibitor, with IC50 values of 0.002, 0.180, 2.85 and 2.22 μM against hPDE5, bPDE6, bPDE1 and hPDE3, respectively. PDE5-IN-15 has good oral bioavailability in dogs. PDE5-IN-15 can be used in research on male erectile dysfunction.
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- CAS No.: 366444-83-9
- Formule: C21H23N5O3
- Masse moléculaire:393.44
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Stockage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Activité biologique
Description
IC50 & Target
[1]|
PDE1 |
PDE5 |
PDE3 |
PDE6 |
Chemical Information
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CAS No. 366444-83-9
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Masse moléculaire 393.44
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Formule C21H23N5O3
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SMILES
COC(C=C12)=CC=C1C=NC=C2CC3=NC(N(C(N(C4=O)C)=O)CC(C)C)=C4N3
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Livraison
Room temperature in continental US; may vary elsewhere.
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Stockage
Please store the product under the recommended conditions in the Certificate of Analysis.
Pureté et documentation
Références
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)