1013098-90-2
1013098-90-2
Chemical Structure
PI3Kα/mTOR-IN-1
- CAS No.: 1013098-90-2
- Formula:C16H18N6O
- Molecular Weight:310.35
IUPAC Name: 2-amino-8-cyclopentyl-4-methyl-6-(1H-pyrazol-4-yl)pyrido[2,3-d]pyrimidin-7(8H)-one
InChIKey: VMGMCPMGGFUNMP-UHFFFAOYSA-N
SMILES: O=C1C(C2=CNN=C2)=CC3=C(C)N=C(N)N=C3N1C4CCCC4
Biological Activity: PI3Kα/mTOR-IN-1 is a potent PI3Kα/mTOR dual inhibitor, with an IC50 of 7 nM for PI3Kα in a cell assay, and Kis of 10.6 nM and 12.5 nM for mTOR and PI3Kα in a cell free assay , respectively.
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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PI3Kα/mTOR-IN-1 | 99.30% | PI3Kα/mTOR-IN-1 is a potent PI3Kα/mTOR dual inhibitor, with an IC50 of 7 nM for PI3Kα in a cell assay, and Kis of 10.6 nM and 12.5 nM for mTOR and PI3Kα in a cell free assay , respectively. | ||||||||||||||||||||
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Keywords
