1036959-27-9
Chemical Structure
(2R)-Vildagliptin
Synonym(s): (2R)-LAF237; (2R)-NVP-LAF 237
- CAS No.: 1036959-27-9
- Formula:C17H25N3O2
- Molecular Weight:303.40
IUPAC Name: (R)-1-(((1r,3S,5R,7S)-3-hydroxyadamantan-1-yl)glycyl)pyrrolidine-2-carbonitrile
InChIKey: SYOKIDBDQMKNDQ-SSOQLKFYSA-N
SMILES: O[C@@]1(C2)C[C@H]3C[C@H](C[C@]2(NCC(N4[C@@H](C#N)CCC4)=O)C3)C1
Biological Activity: (2R)-Vildagliptin is the isomer of Vildagliptin (HY-14291), and can be used as an experimental control. Vildagliptin (LAF237) is a potent, stable, selective dipeptidyl peptidase IV (DPP-IV) inhibitor with an IC50 of 3.5 nM in human Caco-2 cells. Vildagliptin possesses excellent oral bioavailability and potent antihyperglycemic activity[1].
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(2R)-Vildagliptin | (2R)-Vildagliptin is the isomer of Vildagliptin (HY-14291), and can be used as an experimental control. Vildagliptin (LAF237) is a potent, stable, selective dipeptidyl peptidase IV (DPP-IV) inhibitor with an IC50 of 3.5 nM in human Caco-2 cells. Vildagliptin possesses excellent oral bioavailability and potent antihyperglycemic activity. | |||||||||||||||||||||
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Keywords
