103926-64-3
103926-64-3
Chemical Structure
Sepimostat
Synonym(s): FUT-187 free base
- CAS No.: 103926-64-3
- Formula:C21H19N5O2
- Molecular Weight:373.41
IUPAC Name: 6-carbamimidoylnaphthalen-2-yl 4-((4,5-dihydro-1H-imidazol-2-yl)amino)benzoate
InChIKey: QMRJOIUGPCVZPH-UHFFFAOYSA-N
SMILES: O=C(OC1=CC=C2C=C(C(N)=N)C=CC2=C1)C3=CC=C(NC4=NCCN4)C=C3
Biological Activity: Sepimostat (FUT-187 free base) exhibits neuroprotective activity via NR2B N-methyl-D-aspartate receptor antagonism at the Ifenprodil-binding site of the NR2B subunit. Sepimostat inhibits the Ifenprodil binding with a Ki value of 27.7?μM[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Sepimostat | 95.09% | Sepimostat (FUT-187 free base) exhibits neuroprotective activity via NR2B N-methyl-D-aspartate receptor antagonism at the Ifenprodil-binding site of the NR2B subunit. Sepimostat inhibits the Ifenprodil binding with a Ki value of 27.7?μM. | ||||||||||||||||||||
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Sepimostat (Standard) | ≥98% | Sepimostat (Standard) is the analytical standard of Sepimostat. This product is intended for research and analytical applications. Sepimostat (FUT-187 free base) exhibits neuroprotective activity via NR2B N-methyl-D-aspartate receptor antagonism at the Ifenprodil-binding site of the NR2B subunit. Sepimostat inhibits the Ifenprodil binding with a Ki value of 27.7 μM. | ||||||||||||||||||||
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References
Keywords
