114869-83-9
Chemical Structure
Carvedilol Glucuronide
- CAS. Nr.: 114869-83-9
- Formula:C30H34N2O10
- Molecular Weight:582.60
IUPAC Name: (2S,3S,4S,5R,6R)-6-((1-((9H-carbazol-4-yl)oxy)-3-((2-(2-methoxyphenoxy)ethyl)amino)propan-2-yl)oxy)-3,4,5-trihydroxytetrahydro-2H-pyran-2-carboxylic acid
InChIKey: PUVQFGCELBOSRN-VKTJNCFWSA-N
SMILES: OC([C@@H](O[C@H]1OC(COC2=C3C4=CC=CC=C4NC3=CC=C2)CNCCOC5=C(OC)C=CC=C5)[C@@H](O)[C@H](O)[C@H]1O)=O
Biological Activity: Carvedilol Glucuronide is the metabolite of Carvedilol (HY-B0006). Carvedilol (BM 14190) is an antagonist for β/α-1 adrenergic receptor. Carvedilol inhibits lipid peroxidation with an IC50 of 5 μM. Carvedilol is an antihypertensive agent with potential use in angina and congestive heart failure. Carvedilol is an autophagy inducer that inhibits the NLRP3 inflammasome[1].
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Carvedilol Glucuronide | Carvedilol Glucuronide is the metabolite of Carvedilol (HY-B0006). Carvedilol (BM 14190) is an antagonist for β/α-1 adrenergic receptor. Carvedilol inhibits lipid peroxidation with an IC50 of 5 μM. Carvedilol is an antihypertensive agent with potential use in angina and congestive heart failure. Carvedilol is an autophagy inducer that inhibits the NLRP3 inflammasome. | |||||||||||||||||||||
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Keywords
