1222513-26-9
Chemical Structure
CID44216842
Synonym(s): Cdc42-IN-1
- CAS No.: 1222513-26-9
- Formula:C22H20BrN3O3S
- Molecular Weight:486.38
IUPAC Name: 4-(5-(4-bromophenyl)-3-(3-methoxyphenyl)-4,5-dihydro-1H-pyrazol-1-yl)benzenesulfonamide
InChIKey: LPUYDLXQQMWRLR-UHFFFAOYSA-N
SMILES: O=S(C1=CC=C(N2N=C(C3=CC=CC(OC)=C3)CC2C4=CC=C(Br)C=C4)C=C1)(N)=O
Biological Activity: CID44216842 (Cdc42-IN-1) is a potent Cdc42-selective guanine nucleotide binding lead inhibitor. The EC50s for Cdc42 WT and Cdc42Q61L mutant are 1.0 and 1.2 μM in GTP binding assay, respectively. The EC50s for Cdc42 WT and Cdc42Q61L mutant are 0.3 and 0.5 μM in GDP binding assay, respectively. Use as a molecular probe[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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CID44216842 | 99.84% | CID44216842 (Cdc42-IN-1) is a potent Cdc42-selective guanine nucleotide binding lead inhibitor. The EC50s for Cdc42 WT and Cdc42Q61L mutant are 1.0 and 1.2 μM in GTP binding assay, respectively. The EC50s for Cdc42 WT and Cdc42Q61L mutant are 0.3 and 0.5 μM in GDP binding assay, respectively. Use as a molecular probe. | ||||||||||||||||||||
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Keywords
