1233923-95-9

A457 Chemical Structure
1233923-95-9

Chemical Structure

A457

  • CAS No.: 1233923-95-9
  • Formula:C26H33ClN2O3
  • Molecular Weight:457.00

IUPAC Name: 1-benzyl-N-((9-chloro-3,4-dihydro-2H-benzo[b][1,4]dioxepin-7-yl)methyl)-N-isobutylpyrrolidine-3-carboxamide

InChIKey: IOXBZEKQVLIIQH-UHFFFAOYSA-N

SMILES: O=C(N(CC(C)C)CC1=CC(Cl)=C2OCCCOC2=C1)C3CN(CC3)CC4=CC=CC=C4

Biological Activity: A457 is a prokineticin receptor PKR2 antagonist, with an IC50 of 102 nM. A457 can rescue the cell surface expression and function of P290S PKR2, but not W178S and G234D PKR2[1].

Cat. No. Product Name Purity Description Pricing
HY-129317 		A457 A457 is a prokineticin receptor PKR2 antagonist, with an IC50 of 102 nM. A457 can rescue the cell surface expression and function of P290S PKR2, but not W178S and G234D PKR2.
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