1338575-38-4
1338575-38-4
Chemical Structure
FAAH-IN-5
- CAS No.: 1338575-38-4
- Formula:C21H19N3O6S
- Molecular Weight:441.46
IUPAC Name: methyl 5-(hydroxymethyl)furan-2-carboxylate
InChIKey: AZYXDFXRWCDJIZ-UHFFFAOYSA-N
SMILES: O=C(N1CCN(CC1)S(=O)(C2=CC=C3C=CC=CC3=C2)=O)OC4=CC=C(C=C4)[N+]([O-])=O
Biological Activity: FAAH-IN-5 is a dual FAAH/MAGL inhibitor with IC50 values of 0.0105 μM and 0.284 μM, respectively. FAAH-IN-5 shows reduced PAMPA permeability. FAAH-IN-5 produces near-complete blockade of TAMRA-FP labeling of human FAAH and MAGL, and produces significant blockade in homogenates. FAAH-IN-5 can be used in research related to FAAH-mediated diseases[1].
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FAAH-IN-5 | FAAH-IN-5 is a dual FAAH/MAGL inhibitor with IC50 values of 0.0105 μM and 0.284 μM, respectively. FAAH-IN-5 shows reduced PAMPA permeability. FAAH-IN-5 produces near-complete blockade of TAMRA-FP labeling of human FAAH and MAGL, and produces significant blockade in homogenates. FAAH-IN-5 can be used in research related to FAAH-mediated diseases. | |||||||||||||||||||||
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