1345410-31-2
Chemical Structure
Reldesemtiv
Synonym(s): CK-2127107
- CAS No.: 1345410-31-2
- Formula:C19H18F2N6O
- Molecular Weight:384.38
IUPAC Name: 1-(2-((((1r,3r)-3-fluoro-1-(3-fluoropyridin-2-yl)cyclobutyl)methyl)amino)pyrimidin-5-yl)-1H-pyrrole-3-carboxamide
InChIKey: MQXWPWOCXGARRK-HJGJAMNPSA-N
SMILES: O=C(C1=CN(C2=CN=C(NC[C@]3(C4=NC=CC=C4F)C[C@H](F)C3)N=C2)C=C1)N
Biological Activity: Reldesemtiv (CK-2127107) is a selective, orally active and next-generation fast skeletal muscle troponin activator (FSTA). Reldesemtiv selectively activates fast skeletal myofibrils with an EC50 of 3.4 μM. Reldesemtiv increases exercise performance in a heart failure model[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
Reldesemtiv | 99.63% | Reldesemtiv (CK-2127107) is a selective, orally active and next-generation fast skeletal muscle troponin activator (FSTA). Reldesemtiv selectively activates fast skeletal myofibrils with an EC50 of 3.4 μM. Reldesemtiv increases exercise performance in a heart failure model. | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
|
|
Reldesemtiv (Standard) | ≥98% | Reldesemtiv (Standard) is the analytical standard of Reldesemtiv (HY-109121). This product is intended for research and analytical applications. Reldesemtiv (CK-2127107) is a selective, orally active and next-generation fast skeletal muscle troponin activator (FSTA). Reldesemtiv selectively activates fast skeletal myofibrils with an EC50 of 3.4 μM. Reldesemtiv increases exercise performance in a heart failure model. | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
Keywords
