135307-33-4

GW549390X Chemical Structure
135307-33-4

Chemical Structure

GW549390X

  • CAS No.: 135307-33-4
  • Formula:C15H12N2O
  • Molecular Weight:236.27

InChIKey: HFICAVMUTYFODG-UHFFFAOYSA-N

SMILES: C1(NC2=NC=C(C3=CC=CC=C3)O2)=CC=CC=C1

Biological Activity: GW549390X is a dual inhibitor of Fluc and VEGFR2 with IC50 of 0.26 μM and 1.2 μM, respectively. GW549390X can bind to the ATP pocket of FLuc through the aniline side chain and is an ATP-competitive inhibitor of Fluc. GW549390X acts as a protein kinase inhibitor across ATP-dependent and -independent luciferases, with potential implications for Fluc reporter assays[1].

Cat. No. Product Name Purity Description Pricing
HY-160687 		GW549390X GW549390X is a dual inhibitor of Fluc and VEGFR2 with IC50 of 0.26 μM and 1.2 μM, respectively. GW549390X can bind to the ATP pocket of FLuc through the aniline side chain and is an ATP-competitive inhibitor of Fluc. GW549390X acts as a protein kinase inhibitor across ATP-dependent and -independent luciferases, with potential implications for Fluc reporter assays.
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