136013-69-9
136013-69-9
Chemical Structure
WAY-100289
- CAS No.: 136013-69-9
- Formula:C20H27N3O3
- Molecular Weight:357.45
IUPAC Name: 2-(cyclopropylmethoxy)-N-(((1R,3r,5S)-8-methyl-8-azabicyclo[3.2.1]octan-3-yl)carbamoyl)benzamide
InChIKey: VFRIHPWRNNTKEX-MUJYYYPQSA-N
SMILES: O=C(NC(N[C@@H]1C[C@@H](N2C)CC[C@@H]2C1)=O)C3=CC=CC=C3OCC4CC4
Biological Activity: WAY-100289 is an orally active antagonist for 5-HT3 receptor, that exhibits high affinity to the isolated rat vagus nerves with pA2 of 8.9. WAY-100289 inhibits the Bezold-Jarisch reflex in anesthetized and awake rats[1].
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WAY-100289 | WAY-100289 is an orally active antagonist for 5-HT3 receptor, that exhibits high affinity to the isolated rat vagus nerves with pA2 of 8.9. WAY-100289 inhibits the Bezold-Jarisch reflex in anesthetized and awake rats. | |||||||||||||||||||||
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