1426208-69-6
1426208-69-6
Chemical Structure
MGAT2-IN-5
- CAS No.: 1426208-69-6
- Formula:C22H27NO2S2
- Molecular Weight:401.59
IUPAC Name: 6-((4,4-bis(3-methylthiophen-2-yl)but-3-en-1-yl)(methyl)amino)cyclohex-1-ene-1-carboxylic acid
InChIKey: MTVVZKYZYJUBSB-UHFFFAOYSA-N
SMILES: O=C(C1=CCCCC1N(CC/C=C(C2=C(C)C=CS2)\C3=C(C)C=CS3)C)O
Biological Activity: MGAT2-IN-5 (Compound 17b) is a selective inhibitor for mouse GABA transit protection subsidity 2 (mGAT2) with an IC50 of 45 μM. MGAT2-IN-5 exhibits anticonvulsive efficacy in audiogenic seizure (AGS) susceptible frings mouse model with an ED50 of 20.4 mg/kg[1].
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MGAT2-IN-5 | MGAT2-IN-5 (Compound 17b) is a selective inhibitor for mouse GABA transit protection subsidity 2 (mGAT2) with an IC50 of 45 μM. MGAT2-IN-5 exhibits anticonvulsive efficacy in audiogenic seizure (AGS) susceptible frings mouse model with an ED50 of 20.4 mg/kg. | |||||||||||||||||||||
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References
Keywords
