155412-88-7
155412-88-7
Chemical Structure
CCK-B Receptor Antagonist 2
- CAS No.: 155412-88-7
- Formula:C27H28N6O3
- Molecular Weight:484.55
IUPAC Name: (R)-1-(3-aminophenyl)-3-(1-(3,3-dimethyl-2-oxobutyl)-2-oxo-5-(pyridin-2-yl)-2,3-dihydro-1H-benzo[e][1,4]diazepin-3-yl)urea
InChIKey: ABJHMASUFPDZRW-DEOSSOPVSA-N
SMILES: O=C(N[C@H]1C(N(CC(C(C)(C)C)=O)C2=CC=CC=C2C(C3=NC=CC=C3)=N1)=O)NC4=CC=CC(N)=C4
Biological Activity: CCK-B Receptor Antagonist 2, compound 15b, is a potent and orally active Gastrin/CCK-B antagonist with an IC50 value of 0.43 nM. CCK-B Receptor Antagonist 2 also inhibits gastrin/CCK-A activity with an IC50 of 1.82 μM[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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CCK-B Receptor Antagonist 2 | 98.84% | CCK-B Receptor Antagonist 2, compound 15b, is a potent and orally active Gastrin/CCK-B antagonist with an IC50 value of 0.43 nM. CCK-B Receptor Antagonist 2 also inhibits gastrin/CCK-A activity with an IC50 of 1.82 μM. | ||||||||||||||||||||
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References
Keywords
