156001-18-2
Chemical Structure
Embusartan
Synonym(s): BAY 10-6734
- CAS No.: 156001-18-2
- Formula:C25H24FN5O3
- Molecular Weight:461.49
IUPAC Name: methyl 6-butyl-1-((3-fluoro-2'-(1H-tetrazol-5-yl)-[1,1'-biphenyl]-4-yl)methyl)-2-oxo-1,2-dihydropyridine-4-carboxylate
InChIKey: LYVGOAYMIAQLHI-UHFFFAOYSA-N
SMILES: O=C(C(C=C(CCCC)N1CC2=CC=C(C3=CC=CC=C3C4=NN=NN4)C=C2F)=CC1=O)OC
Biological Activity: Embusartan (BAY 10-6734) is a brain-penetrant and effective AT1 receptor blocker. Embusartan inhibits Ang II binding to brain AT1 receptors in the nuclei of central nervous system (CNS) inside due to high lipophilic character. Embusartan is promising for research of sympathetic hyperactivity and hypertension[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
Embusartan | Embusartan (BAY 10-6734) is a brain-penetrant and effective AT1 receptor blocker. Embusartan inhibits Ang II binding to brain AT1 receptors in the nuclei of central nervous system (CNS) inside due to high lipophilic character. Embusartan is promising for research of sympathetic hyperactivity and hypertension. | |||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
Keywords
