1621436-41-6
1621436-41-6
Chemical Structure
Tigolaner
Synonym(s): BAY-1272858
- CAS No.: 1621436-41-6
- Formula:C21H13ClF8N6O
- Molecular Weight:552.81
IUPAC Name: 2-chloro-N-(1-cyanocyclopropyl)-5-(2'-methyl-5'-(perfluoroethyl)-4'-(trifluoromethyl)-2'H-[1,3'-bipyrazol]-4-yl)benzamide
InChIKey: TVAJZOVLQZNNCJ-UHFFFAOYSA-N
SMILES: FC(F)(C(C(C(F)(F)C(F)(F)F)=N1)=C(N2C=C(C(C=C3)=CC(C(NC4(CC4)C#N)=O)=C3Cl)C=N2)N1C)F
Biological Activity: Tigolaner (BAY-1272858) acts on γ-aminobutyric acid (GABA) and glutamate-gated chloride channels. Tigolaner has antiparasitic activity[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Tigolaner | 99.37% | Tigolaner (BAY-1272858) acts on γ-aminobutyric acid (GABA) and glutamate-gated chloride channels. Tigolaner has antiparasitic activity. | ||||||||||||||||||||
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Tigolaner (Standard) | ≥98% | Tigolaner (Standard) is the analytical standard of Tigolaner (HY-109077). This product is intended for research and analytical applications. Tigolaner (BAY-1272858) acts on γ-aminobutyric acid (GABA) and glutamate-gated chloride channels. Tigolaner has antiparasitic activity. | ||||||||||||||||||||
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Tigolaner-d4 | Tigolaner-d4 is deuterium labeled Tigolaner. Tigolaner (BAY-1272858) acts on γ-aminobutyric acid (GABA) and glutamate-gated chloride channels. Tigolaner has antiparasitic activity. | |||||||||||||||||||||
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References
- [1]. Mencke N, et al. Plasma pharmacokinetics of tigolaner, emodepside, and praziquantel following topical administration of a combination product (Felpreva®) and of intravenous administration of the individual active ingredients in cats. Curr Res Parasitol Vector Borne Dis. 2023 Jun 22;4:100126. [Content Brief]
