1628214-07-2
1628214-07-2
Chemical Structure
CPI-4203
- CAS No.: 1628214-07-2
- Formula:C16H14N4O
- Molecular Weight:278.31
IUPAC Name: 6-ethyl-7-oxo-5-(o-tolyl)-4,7-dihydropyrazolo[1,5-a]pyrimidine-3-carbonitrile
InChIKey: OXELDRCVUWWSFZ-UHFFFAOYSA-N
SMILES: N#CC1=C(N2N=C1)NC(C3=C(C=CC=C3)C)=C(C2=O)CC
Biological Activity: CPI-4203 is a potent KDM5A inhibitor with an IC50 of 250 nM. CPI-4203 is competitive with 2-oxoglutarate (2-OG). CPI-4203 is structurally related to CPI-455 (HY-100421) but is less potent[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|---|
|
|
CPI-4203 | 99.0% | CPI-4203 is a potent KDM5A inhibitor with an IC50 of 250 nM. CPI-4203 is competitive with 2-oxoglutarate (2-OG). CPI-4203 is structurally related to CPI-455 (HY-100421) but is less potent. | ||||||||||||||||||||
|
loading...
/
|
|||||||||||||||||||||||
References
Keywords
