CPI-4203
Based on 1 Customer Validation
CPI-4203 is a potent KDM5A inhibitor with an IC50 of 250 nM. CPI-4203 is competitive with 2-oxoglutarate (2-OG). CPI-4203 is structurally related to CPI-455 (HY-100421) but is less potent.
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- Purity: 99.0%
- CAS No.: 1628214-07-2
- 화학식: C16H14N4O
- 분자량:278.31
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보관:Powder -20°C, 3 years ; In solvent -80°C, 6 months , -20°C, 1 month
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
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용액&용해도
- 순도&문서
- References
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Help & FAQs
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Bioactive Compound Library Max
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MCE Bioactive Compound Library
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Bioactive Compound Library
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Methylation Compound Library
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High-Throughput Bioactive Compound Library
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Posttranslational Modification Library
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Biological Activity
IC50: 250 nM (KDM5A)[1]
Chemical Information
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CAS No. 1628214-07-2
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Appearance Solid
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분자량 278.31
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화학식 C16H14N4O
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Color White to off-white
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SMILES
N#CC1=C(N2N=C1)NC(C3=C(C=CC=C3)C)=C(C2=O)CC
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선적
Room temperature in continental US; may vary elsewhere.
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보관
Powder -20°C 3 years In solvent -80°C 6 months -20°C 1 month
용액&용해도
DMSO : 25 mg/mL (89.83 mM; Need ultrasonic and warming; Hygroscopic DMSO has a significant impact on the solubility of product, please use newly opened DMSO)
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
순도&문서
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Data Sheet (274 KB)
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SDS (251 KB)
- English - EN (251 KB)
- Français - FR (251 KB)
- Deutsch - DE (251 KB)
- Norwegian - NO (251 KB)
- Español - ES (251 KB)
- Swedish - SV (251 KB)
- Italian - IT (251 KB)
- Korean - KR (251 KB)
- Portuguese - PT (251 KB)
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Handling Instructions (2659 KB)
References
Complete Stock Solution Preparation Table
Please refer to the solubility information to select the appropriate solvent. Once prepared, please aliquot and store the solution to prevent product inactivation from repeated freeze-thaw cycles.
Storage method and period of stock solution: -80°C, 6 months; -20°C, 1 month. When stored at -80°C, please use it within 6 months. When stored at -20°C, please use it within 1 month.
| Optional Solvent | Concentration Solvent Mass | 1 mg | 5 mg | 10 mg | 25 mg |
|---|---|---|---|---|---|
| DMSO | 1 mM | 3.5931 mL | 17.9656 mL | 35.9312 mL | 89.8279 mL |
| 5 mM | 0.7186 mL | 3.5931 mL | 7.1862 mL | 17.9656 mL | |
| 10 mM | 0.3593 mL | 1.7966 mL | 3.5931 mL | 8.9828 mL | |
| 15 mM | 0.2395 mL | 1.1977 mL | 2.3954 mL | 5.9885 mL | |
| 20 mM | 0.1797 mL | 0.8983 mL | 1.7966 mL | 4.4914 mL | |
| 25 mM | 0.1437 mL | 0.7186 mL | 1.4372 mL | 3.5931 mL | |
| 30 mM | 0.1198 mL | 0.5989 mL | 1.1977 mL | 2.9943 mL | |
| 40 mM | 0.0898 mL | 0.4491 mL | 0.8983 mL | 2.2457 mL | |
| 50 mM | 0.0719 mL | 0.3593 mL | 0.7186 mL | 1.7966 mL | |
| 60 mM | 0.0599 mL | 0.2994 mL | 0.5989 mL | 1.4971 mL | |
| 80 mM | 0.0449 mL | 0.2246 mL | 0.4491 mL | 1.1228 mL |
CPI-4203 Related Classifications
HY-123419 Related Classifications
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