1643958-89-7
1643958-89-7
Chemical Structure
PDK1-IN-RS2
- CAS No.: 1643958-89-7
- Formula:C15H9ClN2O2S3
- Molecular Weight:380.89
IUPAC Name: N-(6-chlorobenzo[d]thiazol-2-yl)benzo[b]thiophene-2-sulfonamide
InChIKey: MZAVPBQCWWIYEQ-UHFFFAOYSA-N
SMILES: O=S(C1=CC2=CC=CC=C2S1)(NC3=NC4=CC=C(C=C4S3)Cl)=O
Biological Activity: PDK1-IN-RS2 is a mimic of peptide docking motif (PIFtide) and is a substrate-selective PDK1 inhibitor with a Kd of 9 μM. PDK1-IN-RS2 suppresses the activation of the downstream kinases S6K1 by PDK1[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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PDK1-IN-RS2 | 98.49% | PDK1-IN-RS2 is a mimic of peptide docking motif (PIFtide) and is a substrate-selective PDK1 inhibitor with a Kd of 9 μM. PDK1-IN-RS2 suppresses the activation of the downstream kinases S6K1 by PDK1. | ||||||||||||||||||||
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References
Keywords
