168830-70-4
168830-70-4
Chemical Structure
YM-58790 free base
- CAS No.: 168830-70-4
- Formula:C27H31N3O2
- Molecular Weight:429.55
IUPAC Name: 1-(4-(methylamino)benzyl)piperidin-4-yl benzhydrylcarbamate
InChIKey: YLHJUSKJLHTVJY-UHFFFAOYSA-N
SMILES: O=C(OC1CCN(CC2=CC=C(NC)C=C2)CC1)NC(C3=CC=CC=C3)C4=CC=CC=C4
Biological Activity: YM-58790 free base is a potent antagonist of mAChR. YM-58790 free base binds M1, M2, M3 with Ki values of 28 nM, 260 nM, and 15 nM. YM-58790 free base exhibits potent inhibitory activity on bladder pressuer in reflexly-evoked rhythmic contraction in rats[1].
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YM-58790 free base | YM-58790 free base is a potent antagonist of mAChR. YM-58790 free base binds M1, M2, M3 with Ki values of 28 nM, 260 nM, and 15 nM. YM-58790 free base exhibits potent inhibitory activity on bladder pressuer in reflexly-evoked rhythmic contraction in rats. | |||||||||||||||||||||
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References
Keywords
