1818234-19-3
1818234-19-3
Chemical Structure
UNC4203
- CAS No.: 1818234-19-3
- Formula:C30H44N6O
- Molecular Weight:504.71
IUPAC Name: (1S,4r)-4-(5-(4-((4-methyl-1,4-diazepan-1-yl)methyl)phenyl)-2-(((S)-pentan-2-yl)amino)-7H-pyrrolo[2,3-d]pyrimidin-7-yl)cyclohexan-1-ol
InChIKey: HYUGTGGDEAGXJP-HRNNMHKYSA-N
SMILES: O[C@@H]1CC[C@H](CC1)N2C=C(C3=CN=C(N=C32)N[C@@H](C)CCC)C4=CC=C(C=C4)CN5CCN(CCC5)C
Biological Activity: UNC4203 is a potent, orally available and highly selective MERTK inhibitor, with IC50s of 1.2 nM, 140 nM, 42 nM and 90 nM for MERTK, AXL, TYRO3 and FLT3, respectively[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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UNC4203 | 99.80% | UNC4203 is a potent, orally available and highly selective MERTK inhibitor, with IC50s of 1.2 nM, 140 nM, 42 nM and 90 nM for MERTK, AXL, TYRO3 and FLT3, respectively. | ||||||||||||||||||||
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References
Keywords
