183173-00-4
Chemical Structure
YM471 free base
- CAS No.: 183173-00-4
- Formula:C39H38F2N4O3
- Molecular Weight:648.74
IUPAC Name: (Z)-N-(4-(5-(2-(4-(dimethylamino)piperidin-1-yl)-2-oxoethylidene)-4,4-difluoro-2,3,4,5-tetrahydro-1H-benzo[b]azepine-1-carbonyl)phenyl)-[1,1'-biphenyl]-2-carboxamide
InChIKey: ICRPTZMWRJGNQI-CLIDGEQKSA-N
SMILES: O=C(C1=CC=C(C=C1)NC(C2=C(C3=CC=CC=C3)C=CC=C2)=O)N4C5=CC=CC=C5/C(C(F)(CC4)F)=C/C(N6CCC(CC6)N(C)C)=O
Biological Activity: YM471 free base is a non-peptide antagonist of vasopressin V1A and V2 receptors with potent and persistent antagonistic activity. YM471 exhibits high affinity for rat V1A and V2 receptors with K values of 0.16 and 0.77 nM, respectively[1].
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YM471 free base | YM471 free base is a non-peptide antagonist of vasopressin V1A and V2 receptors with potent and persistent antagonistic activity. YM471 exhibits high affinity for rat V1A and V2 receptors with K values of 0.16 and 0.77 nM, respectively. | |||||||||||||||||||||
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