1883333-94-5
Chemical Structure
GPR4 antagonist 2
- CAS No.: 1883333-94-5
- Formula:C31H37N5
- Molecular Weight:479.67
IUPAC Name: 2-((2-ethyl-5,7-dimethyl-3H-imidazo[4,5-b]pyridin-3-yl)methyl)-8-(piperidin-1-ylmethyl)-10,11-dihydro-5H-dibenzo[b,f]azepine
InChIKey: YFBWGDXTUXTMEM-UHFFFAOYSA-N
SMILES: N=1C(=CC(=C2N=C(N(C12)CC3=CC=C4NC5=CC=C(C=C5CCC4=C3)CN6CCCCC6)CC)C)C
Biological Activity: GPR4 antagonist 2 is a selective GPR4 antagonist with an IC50 of 67 nM. GPR4 antagonist 2 inhibits pH-dependent GPR4 activation and CRE-driven transcriptional activity. GPR4 antagonist 2 prolongs the survival of mice in a myocardial infarction model. GPR4 antagonist 2 can be used for research on myocardial infarction[1].
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GPR4 antagonist 2 | GPR4 antagonist 2 is a selective GPR4 antagonist with an IC50 of 67 nM. GPR4 antagonist 2 inhibits pH-dependent GPR4 activation and CRE-driven transcriptional activity. GPR4 antagonist 2 prolongs the survival of mice in a myocardial infarction model. GPR4 antagonist 2 can be used for research on myocardial infarction. | |||||||||||||||||||||
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