189003-92-7
189003-92-7
Chemical Structure
Trelanserin
Synonym(s): SL-650472
- CAS No.: 189003-92-7
- Formula:C24H24FN5O2S
- Molecular Weight:465.54
IUPAC Name: 2-(7-fluoro-2-oxo-4-(2-(4-(thieno[3,2-c]pyridin-4-yl)piperazin-1-yl)ethyl)quinolin-1(2H)-yl)acetamide
InChIKey: JDLYOFUDIKMYBL-UHFFFAOYSA-N
SMILES: O=C(N)CN1C(C=C(CCN2CCN(C3=NC=CC4=C3C=CS4)CC2)C5=C1C=C(F)C=C5)=O
Biological Activity: Trelanserin (SL-650472) is a 5-HT receptor antagonist and also an effective in vitro smooth muscle contraction antagonist, competing against the contractions induced by sumatriptan (HY-B0121B) with a pA2 of 8.17±0.36[1].
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Trelanserin | Trelanserin (SL-650472) is a 5-HT receptor antagonist and also an effective in vitro smooth muscle contraction antagonist, competing against the contractions induced by sumatriptan (HY-B0121B) with a pA2 of 8.17±0.36. | |||||||||||||||||||||
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