Trelanserin
Trelanserin (SL-650472) is a 5-HT receptor antagonist and also an effective in vitro smooth muscle contraction antagonist, competing against the contractions induced by sumatriptan (HY-B0121B) with a pA2 of 8.17±0.36.
For research use only. We do not sell to patients.
- CAS No.: 189003-92-7
- Formula: C24H24FN5O2S
- Molecular Weight:465.54
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
To place orders, for customer services and technical support, please contact: MedChemExpress USA
Tel: 609-228-6898 E-mail: [email protected] [email protected]
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Biological Activity
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Chemical Information
- Purity & Documentation
- References
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Help & FAQs
All 5-HT Receptor Isoforms
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Biological Activity
| NCT Number | Sponsor | Condition | Start Date |
Phase
|
|---|---|---|---|---|
| NCT01329991 | Plexxikon| | 2011-05 | PHASE1 |
Chemical Information
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CAS No. 189003-92-7
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Molecular Weight 465.54
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Formula C24H24FN5O2S
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SMILES
O=C(N)CN1C(C=C(CCN2CCN(C3=NC=CC4=C3C=CS4)CC2)C5=C1C=C(F)C=C5)=O
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Synonyms
SL-650472
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)
Trelanserin Related Classifications
HY-14757 Related Classifications
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