1952264-33-3
1952264-33-3
Chemical Structure
ZEN-3862
- CAS No.: 1952264-33-3
- Formula:C19H17FN2O3
- Molecular Weight:340.35
IUPAC Name: 5-(3,5-dimethylisoxazol-4-yl)-1-(3-fluoro-4-(oxiran-2-yl)benzyl)pyridin-2(1H)-one
InChIKey: VQHDSZCBMWYGEK-UHFFFAOYSA-N
SMILES: O=C(C=CC(C1=C(C)ON=C1C)=C2)N2CC3=CC(F)=C(C4OC4)C=C3
Biological Activity: ZEN-3862 is a BET inhibitor with IC50s of 0.16 and 0.13 μM for BRD4(BD1) and BRD4(BD2) , respectively. ZEN-3862 can be used to form PROTACs to induce degradation of BRD4[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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ZEN-3862 | 98.86% | ZEN-3862 is a BET inhibitor with IC50s of 0.16 and 0.13 μM for BRD4(BD1) and BRD4(BD2) , respectively. ZEN-3862 can be used to form PROTACs to induce degradation of BRD4. | ||||||||||||||||||||
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References
Keywords
