2095719-90-5
2095719-90-5
Chemical Structure
ERK1/2 inhibitor 1
- CAS No.: 2095719-90-5
- Formula:C29H32ClN5O4
- Molecular Weight:550.05
IUPAC Name: (R)-2-(6-(5-chloro-2-((tetrahydro-2H-pyran-4-yl)amino)pyrimidin-4-yl)-1-oxoisoindolin-2-yl)-N-((S)-2-hydroxy-1-(m-tolyl)ethyl)propanamide
InChIKey: XHOJEECXVUMYMF-IQGLISFBSA-N
SMILES: ClC1=CN=C(NC2CCOCC2)N=C1C3=CC=C(CN([C@H](C)C(N[C@H](CO)C4=CC=CC(C)=C4)=O)C5=O)C5=C3
Biological Activity: ERK1/2 inhibitor 1 is a potent, orally bioavailable ERK1/2 inhibitor, showing 60% inhibition at 1 nM and an IC50 of 3.0 nM against ERK1 and ERK2, respectively[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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ERK1/2 inhibitor 1 | 99.58% | ERK1/2 inhibitor 1 is a potent, orally bioavailable ERK1/2 inhibitor, showing 60% inhibition at 1 nM and an IC50 of 3.0 nM against ERK1 and ERK2, respectively. | ||||||||||||||||||||
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References
Keywords
