216853-60-0
216853-60-0
Chemical Structure
NS3861 fumarate
- CAS No.: 216853-60-0
- Formula:C16H18BrNO4S
- Molecular Weight:400.29
IUPAC Name: 3-(3-bromothiophen-2-yl)-8-methyl-8-azabicyclo[3.2.1]oct-2-ene fumarate
InChIKey: KXBSQPLWTVQFGJ-WLHGVMLRSA-N
SMILES: BrC1=C(C2=CC(CC3)N(C)C3C2)SC=C1.OC(/C=C/C(O)=O)=O
Biological Activity: NS3861 fumarate is an agonist of nicotinic acetylcholine receptors (nAChRs) and binds with high affinity to heteromeric α3β4 nAChR. The binding Ki values of 0.62, 25, 7.8, 55 nM for α3β4, α3β2, α4β4, α4β2, respectively[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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NS3861 fumarate | 99.71% | NS3861 fumarate is an agonist of nicotinic acetylcholine receptors (nAChRs) and binds with high affinity to heteromeric α3β4 nAChR. The binding Ki values of 0.62, 25, 7.8, 55 nM for α3β4, α3β2, α4β4, α4β2, respectively. | ||||||||||||||||||||
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NS3861 fumarate (Standard) | ≥98% | NS3861 fumarate (Standard) is the analytical standard of NS3861 (fumarate) (HY-110121). This product is intended for research and analytical applications. NS3861 fumarate is an agonist of nicotinic acetylcholine receptors (nAChRs) and binds with high affinity to heteromeric α3β4 nAChR. The binding Ki values of 0.62, 25, 7.8, 55 nM for α3β4, α3β2, α4β4, α4β2, respectively. | ||||||||||||||||||||
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References
