2259641-47-7
2259641-47-7
Chemical Structure
Ep300/CREBBP-IN-3
- CAS No.: 2259641-47-7
- Formula:C26H25F4N5O3
- Molecular Weight:531.50
IUPAC Name: (2R,4R)-4-fluoro-N-(1H-pyrazolo[4,3-b]pyridin-5-yl)-1-(1-(4-(2,2,2-trifluoroacetyl)phenyl)cyclohexane-1-carbonyl)pyrrolidine-2-carboxamide
InChIKey: KBEWWRZSPXHLHF-YLJYHZDGSA-N
SMILES: O=C([C@@H]1N(C(C2(C3=CC=C(C(C(F)(F)F)=O)C=C3)CCCCC2)=O)C[C@H](F)C1)NC4=CC=C(NN=C5)C5=N4
Biological Activity: Ep300/CREBBP-IN-3 (Example 61) is a potent Ep300 and CREBBP inhibitor with IC50s of 0.056 and 0.095 μM, respectively. Ep300/CREBBP-IN-3 can be used for the research of cancer[1].
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Ep300/CREBBP-IN-3 | Ep300/CREBBP-IN-3 (Example 61) is a potent Ep300 and CREBBP inhibitor with IC50s of 0.056 and 0.095 μM, respectively. Ep300/CREBBP-IN-3 can be used for the research of cancer. | |||||||||||||||||||||
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References
Keywords
