2374972-35-5
2374972-35-5
Chemical Structure
(R,R)-CPI-1612
- CAS No.: 2374972-35-5
- Formula:C27H26N6O
- Molecular Weight:450.53
IUPAC Name: (R)-2-(((R)-2-(4-cyanophenyl)propyl)amino)-N-(5-(1-methyl-1H-pyrazol-4-yl)pyridin-2-yl)-2-phenylacetamide
InChIKey: SEDFZSHSBUXKAC-AFMDSPMNSA-N
SMILES: CN(N=C1)C=C1C(C=N2)=CC=C2NC([C@@H](C3=CC=CC=C3)NC[C@@H](C4=CC=C(C=C4)C#N)C)=O
Biological Activity: (R,R)-CPI-1612 is the isomer of CPI-1612 (HY-136285), and can be used as an experimental control. CPI-1612 is a highly potent, orally active EP300/CBP histone acetyltransferase (HAT) inhibitor with an IC50 of 8.1 nM for EP300 HAT. CPI-1612 has an anticancer activity[1].
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(R,R)-CPI-1612 | 99.68% | (R,R)-CPI-1612 is the isomer of CPI-1612 (HY-136285), and can be used as an experimental control. CPI-1612 is a highly potent, orally active EP300/CBP histone acetyltransferase (HAT) inhibitor with an IC50 of 8.1 nM for EP300 HAT. CPI-1612 has an anticancer activity. | ||||||||||||||||||||
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