2378640-92-5
2378640-92-5
Chemical Structure
Enpp-1-IN-2
- CAS No.: 2378640-92-5
- Formula:C15H18N6
- Molecular Weight:282.34
IUPAC Name: 6-(3-aminobenzyl)-N,N,5-trimethyl-[1,2,4]triazolo[1,5-a]pyrimidin-7-amine
InChIKey: VUDSCOCEYOZLJD-UHFFFAOYSA-N
SMILES: CC1=NC2=NC=NN2C(N(C)C)=C1CC3=CC=CC(N)=C3
Biological Activity: Enpp-1-IN-2 (Compound C) is a potent ENPP1 (ectonucleotide pyrophosphatase/phosphodiesterase 1) inhibitor with IC50 values of 0.26, 0.48 and 2.0 μM evaluated by means of TG-mAMP, pNP-TMP, and ATP assays, respectively. TG (Tokyo Green)-mAMP: a newly synthesized sensitive ENPP1 fluorescence probe[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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Enpp-1-IN-2 | 99.51% | Enpp-1-IN-2 (Compound C) is a potent ENPP1 (ectonucleotide pyrophosphatase/phosphodiesterase 1) inhibitor with IC50 values of 0.26, 0.48 and 2.0 μM evaluated by means of TG-mAMP, pNP-TMP, and ATP assays, respectively. TG (Tokyo Green)-mAMP: a newly synthesized sensitive ENPP1 fluorescence probe. | ||||||||||||||||||||
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References
Keywords
