2409963-50-2
2409963-50-2
Chemical Structure
PXS-4787
- CAS No.: 2409963-50-2
- Formula:C10H12FNO2S
- Molecular Weight:229.27
IUPAC Name: (Z)-3-fluoro-4-(phenylsulfonyl)but-2-en-1-amine
InChIKey: HTUIHUIRTWMKFB-TWGQIWQCSA-N
SMILES: NC/C=C(CS(=O)(C1=CC=CC=C1)=O)\F
Biological Activity: PXS-4787 is a specific and effective pan-LOX (lysyl oxidase) inhibitor for abolishing lysyl oxidase activity. PXS-4787 inhibits LOX with IC50s of 2 μM (Bovine LOX), 3.2 μM (rh LOXL1), 0.6 μM (rh LOXL2), 1.4 μM (rh LOXL3), 0.2 μM (rh LOXL4), respectively[1].
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PXS-4787 | PXS-4787 is a specific and effective pan-LOX (lysyl oxidase) inhibitor for abolishing lysyl oxidase activity. PXS-4787 inhibits LOX with IC50s of 2 μM (Bovine LOX), 3.2 μM (rh LOXL1), 0.6 μM (rh LOXL2), 1.4 μM (rh LOXL3), 0.2 μM (rh LOXL4), respectively. | |||||||||||||||||||||
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References
Keywords
