2411173-40-3
2411173-40-3
Chemical Structure
EP055
- CAS No.: 2411173-40-3
- Formula:C15H17N7O6S
- Molecular Weight:423.40
InChIKey: BWGDSYILNBRKLQ-UHFFFAOYSA-N
SMILES: O=C(CSC1=NC(NC2=CC=C(C(O)=C2)NC(C)=O)=NC(NNC(OC)=O)=N1)O
Biological Activity: EP055 is a non-hormonal male contraceptive. EP055 targets to sperm protein EPPIN and inhibits anti-EPPIN antibodies from binding EPPIN with an IC50 of 1121 μM. EP055 can inhibit sperm motility (IC50 = 199.5 μM) by reducing the internal pH and Ca2+ levels of the sperm, thereby causing the sperm to aggregate. EP055 can be used for development of male contraceptive[1].
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EP055 | EP055 is a non-hormonal male contraceptive. EP055 targets to sperm protein EPPIN and inhibits anti-EPPIN antibodies from binding EPPIN with an IC50 of 1121 μM. EP055 can inhibit sperm motility (IC50 = 199.5 μM) by reducing the internal pH and Ca2+ levels of the sperm, thereby causing the sperm to aggregate. EP055 can be used for development of male contraceptive. | |||||||||||||||||||||
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References
Keywords
