2413850-54-9
2413850-54-9
Chemical Structure
GABAA receptor modulator-2
- CAS. Nr.: 2413850-54-9
- Formula:C22H22FN3O5S
- Molecular Weight:459.49
IUPAC Name: 1-(2-((3-(4-fluorophenyl)-5-methylisoxazol-4-yl)methoxy)-7,8-dihydro-1,6-naphthyridin-6(5H)-yl)-2-(methylsulfonyl)ethan-1-one
InChIKey: GTVLCHCOKLXHLY-UHFFFAOYSA-N
SMILES: CC1=C(C(C2=CC=C(C=C2)F)=NO1)COC3=NC4=C(C=C3)CN(C(CS(C)(=O)=O)=O)CC4
Biological Activity: GABAA receptor modulator-2 (Compound 20) is selective, orally active α5-GABAAR negative allosteric modulator (NAM) with a Ki of 4.1 nM. GABAA receptor modulator-2 shows high-metabolic stability and good CNS safety[1].
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GABAA receptor modulator-2 | GABAA receptor modulator-2 (Compound 20) is selective, orally active α5-GABAAR negative allosteric modulator (NAM) with a Ki of 4.1 nM. GABAA receptor modulator-2 shows high-metabolic stability and good CNS safety. | |||||||||||||||||||||
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