2556833-08-8
2556833-08-8
Chemical Structure
mGAT-IN-1
- CAS No.: 2556833-08-8
- Formula:C28H34ClN3O2S2
- Molecular Weight:544.17
IUPAC Name: 4-acetamido-2-((4,4-bis(3-methylthiophen-2-yl)but-3-en-1-yl)(methyl)amino)-N-(2-chlorobenzyl)butanamide
InChIKey: BYIMWNNOGMXRCA-UHFFFAOYSA-N
SMILES: CC(NCCC(N(CC/C=C(C1=C(C=CS1)C)/C2=C(C=CS2)C)C)C(NCC3=C(C=CC=C3)Cl)=O)=O
Biological Activity: mGAT-IN-1 (compound 28) is a potent and non-selective GAT inhibitor. mGAT-IN-1 has a high inhibitory potency toward mGAT3, with an IC50 of 2.5 μM and pIC50 of 5.61[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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mGAT-IN-1 | mGAT-IN-1 (compound 28) is a potent and non-selective GAT inhibitor. mGAT-IN-1 has a high inhibitory potency toward mGAT3, with an IC50 of 2.5 μM and pIC50 of 5.61. | |||||||||||||||||||||
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References
Keywords
