mGAT-IN-1
mGAT-IN-1 (compound 28) is a potent and non-selective GAT inhibitor. mGAT-IN-1 has a high inhibitory potency toward mGAT3, with an IC50 of 2.5 μM and pIC50 of 5.61.
For research use only. We do not sell to patients.
- CAS No.: 2556833-08-8
- Formula: C28H34ClN3O2S2
- Molecular Weight:544.17
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Storage:
Please store the product under the recommended conditions in the Certificate of Analysis.
Biological Activity
IC50: 2.5 μM (mGAT3); pIC50: 5.06 ± 0.02 (mGAT1), 5.35 ± 0.08 (mGAT2), 5.61 ± 0.07 (mGAT3), 5.21 ± 0.05 (mGAT4)[1]
Chemical Information
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CAS No. 2556833-08-8
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Molecular Weight 544.17
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Formula C28H34ClN3O2S2
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SMILES
CC(NCCC(N(CC/C=C(C1=C(C=CS1)C)/C2=C(C=CS2)C)C)C(NCC3=C(C=CC=C3)Cl)=O)=O
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Shipping
Room temperature in continental US; may vary elsewhere.
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Storage
Please store the product under the recommended conditions in the Certificate of Analysis.
Purity & Documentation
References
Calculators
Concentration (start) × Volume (start) = Concentration (final) × Volume (final)