2688745-47-1
2688745-47-1
Chemical Structure
Y08284
- CAS No.: 2688745-47-1
- Formula:C26H25FN4O4
- Molecular Weight:476.50
IUPAC Name: (E)-N-methyl-N'-(2-methyl-4-(methyl-d3)phenyl)-N-((E)-((2-methyl-4-(methyl-d3)phenyl)imino)methyl)formimidamide
InChIKey: KKCORLIQMAQULG-UHFFFAOYSA-N
SMILES: O=C(C1=C2C=C(OC)C=CN2C(C(C)=O)=C1)NC3=CC(C(O)C)=CC(C4=CN(C5CC5)N=C4)=C3F
Biological Activity: Y08284 is a potent, selective, oral active CBP bromodomain inhibitor with an IC50 of 4.21 nM. Y08284 suppresses the proliferation of prostate cancer cell lines LNCaP, C4-2B, and 22Rv1. Antitumor activity[1].
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Y08284 | Y08284 is a potent, selective, oral active CBP bromodomain inhibitor with an IC50 of 4.21 nM. Y08284 suppresses the proliferation of prostate cancer cell lines LNCaP, C4-2B, and 22Rv1. Antitumor activity. | |||||||||||||||||||||
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References
Keywords
