2772949-38-7
Chemical Structure
CB1/2 agonist 4
- CAS No.: 2772949-38-7
- Formula:C27H45NO3
- Molecular Weight:431.65
IUPAC Name: N-cyclopropyl-8-(3-methoxy-5-(2-methyloctan-2-yl)phenoxy)octanamide
InChIKey: CWNFRGKJPKDJSQ-UHFFFAOYSA-N
SMILES: O=C(NC1CC1)CCCCCCCOC2=CC(C(CCCCCC)(C)C)=CC(OC)=C2
Biological Activity: CB1/2 agonist 4 is a full CB1 agonist and CB2 partial agonist with EC50 values of 15.09 nM and 1.16 nM, respectively. CB1/2 agonist 4 also has hCB1 and hCB2 receptor affinities with Ki values of 1.1 nM and 4.2 nM, respectively. CB1/2 agonist 4 has a significant antinociceptive activity, and also can activate cannabinoid and TRPV1 receptor with values of IC50 and EC50 is 0.8 μM and 0.12 μM, respectively[1].
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CB1/2 agonist 4 | CB1/2 agonist 4 is a full CB1 agonist and CB2 partial agonist with EC50 values of 15.09 nM and 1.16 nM, respectively. CB1/2 agonist 4 also has hCB1 and hCB2 receptor affinities with Ki values of 1.1 nM and 4.2 nM, respectively. CB1/2 agonist 4 has a significant antinociceptive activity, and also can activate cannabinoid and TRPV1 receptor with values of IC50 and EC50 is 0.8 μM and 0.12 μM, respectively. | |||||||||||||||||||||
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Keywords
