2816062-15-2
2816062-15-2
Chemical Structure
AP-7-168
- CAS No.: 2816062-15-2
- Formula:C20H19BrF2N4
- Molecular Weight:433.29
InChIKey: XPSOVAYWMLKDBS-UHFFFAOYSA-N
SMILES: FC1=C(C=C(C=C1)NC2=NC3=CC=C(C=C3C(NC4CCCCC4)=N2)Br)F
Biological Activity: AP-7-168, molecular glues, is a β-arrestin-biased negative allosteric modulator of the β2-adrenergic receptor (β2AR). AP-7-168 can promote β2AR homodimerization and inhibit GRK5-mediated β2AR phosphorylation. AP-7-168 can sustain bronchorelaxation in cell and tissue. AP-7-168 can be used for the researches of inflammation and immunology, such as asthma[1].
| Cat. No. | Product Name | Purity | Description | Pricing | |||||||||||||||||||
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AP-7-168 | 99.89% | AP-7-168, molecular glues, is a β-arrestin-biased negative allosteric modulator of the β2-adrenergic receptor (β2AR). AP-7-168 can promote β2AR homodimerization and inhibit GRK5-mediated β2AR phosphorylation. AP-7-168 can sustain bronchorelaxation in cell and tissue. AP-7-168 can be used for the researches of inflammation and immunology, such as asthma. | ||||||||||||||||||||
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