2848632-52-8
2848632-52-8
Chemical Structure
Antitumor agent-101
- CAS No.: 2848632-52-8
- Formula:C26H38N6O3
- Molecular Weight:482.62
InChIKey: GHCDVBSKNGUGCK-UHFFFAOYSA-N
SMILES: COC1=CC2=C(N=C(N(C)C(C=C)=O)N=C2NC3CCN(C)CC3)C=C1OCCCN4CCCC4
Biological Activity: Antitumor agent-101 is a selective covalent inhibitor of lysine methyltransferases G9a/GLP, with IC50s of 8.5 nM and 5.5 nM for G9a and GLP, respectively. Antitumor agent-101 shows antitumor efficacy in the PANC-1 xenograft model[1].
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Antitumor agent-101 | Antitumor agent-101 is a selective covalent inhibitor of lysine methyltransferases G9a/GLP, with IC50s of 8.5 nM and 5.5 nM for G9a and GLP, respectively. Antitumor agent-101 shows antitumor efficacy in the PANC-1 xenograft model. | |||||||||||||||||||||
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